Assay Detail
Functional
CHEMBL2363459
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SANGER: Inhibition of human NB69 cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NB69 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.89 | 9.24 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.24 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 9.06 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 8.98 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.91 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.61 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.24 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.20 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.09 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 8.02 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.96 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.80 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.65 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.34 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 7.12 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 7.11 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.10 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 7.10 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 6.95 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.87 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 6.84 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 6.79 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.76 |
| CHEMBL2144069 | — | — | 1 | 6.72 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.67 |
| CHEMBL379300 | A-443654 | — | 1 | 6.64 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 6.61 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.57 |
| CHEMBL401930 | — | — | 1 | 6.53 |
| CHEMBL509032 | TAE-684 | — | 1 | 6.50 |
| CHEMBL1256459 | TORIN1 | — | 1 | 6.49 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.5694 | nM | 9.24 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 0.8731 | nM | 9.06 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 1.046 | nM | 8.98 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 1.218 | nM | 8.91 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 2.46 | nM | 8.61 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 5.73 | nM | 8.24 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 6.293 | nM | 8.20 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 8.07 | nM | 8.09 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 9.464 | nM | 8.02 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 11.02 | nM | 7.96 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 15.65 | nM | 7.80 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 22.53 | nM | 7.65 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 45.53 | nM | 7.34 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 75.73 | nM | 7.12 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 78.0 | nM | 7.11 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 79.2 | nM | 7.10 |
| CHEMBL803 | CYTARABINE | IC50 | = | 79.48 | nM | 7.10 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 113.01 | nM | 6.95 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 135.0 | nM | 6.87 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 144.36 | nM | 6.84 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 161.8 | nM | 6.79 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 175.06 | nM | 6.76 |
| CHEMBL2144069 | — | IC50 | = | 191.31 | nM | 6.72 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 212.73 | nM | 6.67 |
| CHEMBL379300 | A-443654 | IC50 | = | 226.69 | nM | 6.64 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 245.27 | nM | 6.61 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 270.87 | nM | 6.57 |
| CHEMBL401930 | — | IC50 | = | 292.78 | nM | 6.53 |
| CHEMBL509032 | TAE-684 | IC50 | = | 317.87 | nM | 6.50 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 321.88 | nM | 6.49 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 363.69 | nM | 6.44 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 411.71 | nM | 6.38 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 414.63 | nM | 6.38 |
| CHEMBL3349342 | — | IC50 | = | 556.88 | nM | 6.25 |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 582.57 | nM | 6.24 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 598.25 | nM | 6.22 |
| CHEMBL939 | GEFITINIB | IC50 | = | 614.35 | nM | 6.21 |
| CHEMBL512504 | — | IC50 | = | 685.75 | nM | 6.16 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 705.49 | nM | 6.15 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 734.67 | nM | 6.13 |
| CHEMBL217354 | — | IC50 | = | 876.72 | nM | 6.06 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 922.54 | nM | 6.04 |
| CHEMBL1173055 | RUCAPARIB | IC50 | = | 945.52 | nM | 6.02 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 1029.45 | nM | 5.99 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 1053.9 | nM | 5.98 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 1087.5 | nM | 5.96 |
| CHEMBL577784 | BX-795 | IC50 | = | 1158.65 | nM | 5.94 |
| CHEMBL513909 | BI-2536 | IC50 | = | 1261.48 | nM | 5.90 |
| CHEMBL217092 | SARACATINIB | IC50 | = | 1374.97 | nM | 5.86 |
| CHEMBL585951 | — | IC50 | = | 1430.83 | nM | 5.84 |