Assay Detail
Functional
CHEMBL2363486
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SANGER: Inhibition of human NCI-H1703 cell growth in a cell viability assay.
82
Total Activities
81
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NCI-H1703 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 82 | 5.87 | 9.04 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 9.04 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.84 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.80 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.55 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.43 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.19 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 8.19 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.11 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.99 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 7.79 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.63 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.50 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 7.30 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.21 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.90 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.71 |
| CHEMBL217354 | — | — | 1 | 6.66 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.56 |
| CHEMBL176544 | — | — | 1 | 6.52 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.46 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.38 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.28 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.23 |
| CHEMBL585951 | — | — | 1 | 6.23 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.15 |
| CHEMBL255863 | NILOTINIB | 4.0 | 1 | 5.92 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 5.89 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.64 |
| CHEMBL2363137 | — | — | 1 | 5.48 |
| CHEMBL288441 | BOSUTINIB | 4.0 | 1 | 5.47 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1289926 | AXITINIB | IC50 | = | 0.9022 | nM | 9.04 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 1.431 | nM | 8.84 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.568 | nM | 8.80 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 2.834 | nM | 8.55 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 3.685 | nM | 8.43 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 6.515 | nM | 8.19 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 6.433 | nM | 8.19 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 7.758 | nM | 8.11 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 10.14 | nM | 7.99 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 16.12 | nM | 7.79 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 23.21 | nM | 7.63 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 31.78 | nM | 7.50 |
| CHEMBL803 | CYTARABINE | IC50 | = | 49.81 | nM | 7.30 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 61.78 | nM | 7.21 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 126.42 | nM | 6.90 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 196.15 | nM | 6.71 |
| CHEMBL217354 | — | IC50 | = | 217.09 | nM | 6.66 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 276.88 | nM | 6.56 |
| CHEMBL176544 | — | IC50 | = | 298.97 | nM | 6.52 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 344.83 | nM | 6.46 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 414.46 | nM | 6.38 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 522.74 | nM | 6.28 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 594.27 | nM | 6.23 |
| CHEMBL585951 | — | IC50 | = | 590.81 | nM | 6.23 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 704.73 | nM | 6.15 |
| CHEMBL255863 | NILOTINIB | IC50 | = | 1188.7 | nM | 5.92 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 1299.39 | nM | 5.89 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 2297.23 | nM | 5.64 |
| CHEMBL2363137 | — | IC50 | = | 3287.24 | nM | 5.48 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 3418.12 | nM | 5.47 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 5358.26 | nM | 5.27 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 9343.75 | nM | 5.03 |
| CHEMBL105442 | CI-1040 | IC50 | = | 12261.58 | nM | 4.91 |
| CHEMBL258844 | — | IC50 | = | 15577.01 | nM | 4.81 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 16592.64 | nM | 4.78 |
| CHEMBL221137 | EMBELIN | IC50 | = | 19086.0 | nM | 4.72 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 20308.77 | nM | 4.69 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 20431.77 | nM | 4.69 |
| CHEMBL573107 | — | IC50 | = | 20817.29 | nM | 4.68 |
| CHEMBL135561 | — | IC50 | = | 24152.74 | nM | 4.62 |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 26459.33 | nM | 4.58 |
| CHEMBL191384 | — | IC50 | = | 27694.78 | nM | 4.56 |
| CHEMBL103667 | DORAMAPIMOD | IC50 | = | 28041.26 | nM | 4.55 |
| CHEMBL188678 | — | IC50 | = | 31090.49 | nM | 4.51 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 35173.92 | nM | 4.45 |
| CHEMBL399530 | — | IC50 | = | 36942.85 | nM | 4.43 |
| CHEMBL512504 | — | IC50 | = | 39561.8 | nM | 4.40 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 46059.22 | nM | 4.34 |
| CHEMBL939 | GEFITINIB | IC50 | = | 48335.2 | nM | 4.32 |
| CHEMBL1230020 | PLX-4720 | IC50 | = | 52242.12 | nM | 4.28 |