Assay Detail
Functional
CHEMBL2363570
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SANGER: Inhibition of human OE19 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | OE19 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.29 | 8.33 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.33 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.25 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.88 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.71 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 7.51 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.44 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.70 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 6.47 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.44 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 6.38 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.22 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 6.15 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.09 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.00 |
| CHEMBL585951 | — | — | 1 | 5.96 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 5.81 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 5.78 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 5.77 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 5.73 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 5.67 |
| CHEMBL191384 | — | — | 1 | 5.53 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 5.49 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 5.48 |
| CHEMBL2363137 | — | — | 1 | 5.42 |
| CHEMBL412142 | LADUVIGLUSIB | 1.0 | 1 | 5.40 |
| CHEMBL1084546 | PF-00562271 | 1.0 | 1 | 5.33 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 5.26 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 5.25 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 5.24 |
| CHEMBL217354 | — | — | 1 | 5.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 4.661 | nM | 8.33 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 5.591 | nM | 8.25 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 13.24 | nM | 7.88 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 19.5 | nM | 7.71 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 30.77 | nM | 7.51 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 36.52 | nM | 7.44 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 200.18 | nM | 6.70 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 340.53 | nM | 6.47 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 364.96 | nM | 6.44 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 412.2 | nM | 6.38 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 596.48 | nM | 6.22 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 702.16 | nM | 6.15 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 807.34 | nM | 6.09 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 1010.75 | nM | 6.00 |
| CHEMBL585951 | — | IC50 | = | 1099.44 | nM | 5.96 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 1544.6 | nM | 5.81 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 1655.18 | nM | 5.78 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 1715.12 | nM | 5.77 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1877.07 | nM | 5.73 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 2143.52 | nM | 5.67 |
| CHEMBL191384 | — | IC50 | = | 2922.1 | nM | 5.53 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 3273.33 | nM | 5.49 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 3284.89 | nM | 5.48 |
| CHEMBL2363137 | — | IC50 | = | 3777.01 | nM | 5.42 |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 3964.51 | nM | 5.40 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 4631.45 | nM | 5.33 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 5517.21 | nM | 5.26 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 5686.24 | nM | 5.25 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 5754.09 | nM | 5.24 |
| CHEMBL217354 | — | IC50 | = | 5977.55 | nM | 5.22 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 7655.03 | nM | 5.12 |
| CHEMBL258844 | — | IC50 | = | 7766.84 | nM | 5.11 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 8762.62 | nM | 5.06 |
| CHEMBL1190711 | — | IC50 | = | 8900.46 | nM | 5.05 |
| CHEMBL2134202 | — | IC50 | = | 10173.34 | nM | 4.99 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 11551.17 | nM | 4.94 |
| CHEMBL939 | GEFITINIB | IC50 | = | 11936.73 | nM | 4.92 |
| CHEMBL259181 | — | IC50 | = | 11910.95 | nM | 4.92 |
| CHEMBL3349342 | — | IC50 | = | 14060.89 | nM | 4.85 |
| CHEMBL573107 | — | IC50 | = | 14007.45 | nM | 4.85 |
| CHEMBL477989 | SB590885 | IC50 | = | 14123.85 | nM | 4.85 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 15154.11 | nM | 4.82 |
| CHEMBL202721 | — | IC50 | = | 15231.02 | nM | 4.82 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 16517.56 | nM | 4.78 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 16524.0 | nM | 4.78 |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 18329.72 | nM | 4.74 |
| CHEMBL135561 | — | IC50 | = | 22283.18 | nM | 4.65 |
| CHEMBL803 | CYTARABINE | IC50 | = | 22440.11 | nM | 4.65 |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 26215.27 | nM | 4.58 |
| CHEMBL399530 | — | IC50 | = | 28786.23 | nM | 4.54 |