Assay Detail
Functional
CHEMBL2363593
Review assay metadata, readout intent, target linkage, and publication context from the same page.
SANGER: Inhibition of human QIMR-WIL cell growth in a cell viability assay.
130
Total Activities
129
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | QIMR-WIL |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 130 | 5.89 | 9.11 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.11 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 9.05 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.93 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.52 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.36 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 8.24 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.05 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.99 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 7.93 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.90 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 7.79 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.68 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.51 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.48 |
| CHEMBL512504 | — | — | 1 | 7.44 |
| CHEMBL514499 | GW843682X | — | 1 | 7.37 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 7.37 |
| CHEMBL300389 | — | — | 1 | 7.31 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.09 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 7.03 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.92 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.88 |
| CHEMBL379975 | — | — | 1 | 6.87 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 6.86 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.81 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.79 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.74 |
| CHEMBL379300 | A-443654 | — | 1 | 6.59 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 6.57 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.48 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.7753 | nM | 9.11 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 0.8888 | nM | 9.05 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 1.186 | nM | 8.93 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 3.043 | nM | 8.52 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 4.381 | nM | 8.36 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 5.708 | nM | 8.24 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 8.95 | nM | 8.05 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 10.33 | nM | 7.99 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 11.85 | nM | 7.93 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 12.69 | nM | 7.90 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 16.31 | nM | 7.79 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 20.72 | nM | 7.68 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 30.6 | nM | 7.51 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 32.93 | nM | 7.48 |
| CHEMBL512504 | — | IC50 | = | 36.42 | nM | 7.44 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 42.87 | nM | 7.37 |
| CHEMBL514499 | GW843682X | IC50 | = | 42.33 | nM | 7.37 |
| CHEMBL300389 | — | IC50 | = | 48.85 | nM | 7.31 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 80.55 | nM | 7.09 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 94.09 | nM | 7.03 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 119.58 | nM | 6.92 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 132.23 | nM | 6.88 |
| CHEMBL379975 | — | IC50 | = | 134.99 | nM | 6.87 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 139.41 | nM | 6.86 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 154.58 | nM | 6.81 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 163.11 | nM | 6.79 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 181.89 | nM | 6.74 |
| CHEMBL379300 | A-443654 | IC50 | = | 256.47 | nM | 6.59 |
| CHEMBL513909 | BI-2536 | IC50 | = | 271.55 | nM | 6.57 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 334.24 | nM | 6.48 |
| CHEMBL585951 | — | IC50 | = | 343.43 | nM | 6.46 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 430.49 | nM | 6.37 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 426.76 | nM | 6.37 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 451.5 | nM | 6.34 |
| CHEMBL220241 | GSK-269962A | IC50 | = | 490.04 | nM | 6.31 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 527.33 | nM | 6.28 |
| CHEMBL1190711 | — | IC50 | = | 581.8 | nM | 6.24 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 636.56 | nM | 6.20 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 683.43 | nM | 6.17 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 706.29 | nM | 6.15 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 851.41 | nM | 6.07 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 865.2 | nM | 6.06 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 862.03 | nM | 6.06 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 1090.58 | nM | 5.96 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 1131.34 | nM | 5.95 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 1343.84 | nM | 5.87 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 1491.16 | nM | 5.83 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 1554.2 | nM | 5.81 |
| CHEMBL191334 | NUTLIN-3 | IC50 | = | 1608.54 | nM | 5.79 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 1653.64 | nM | 5.78 |