Assay Detail
Functional
CHEMBL2363658
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SANGER: Inhibition of human SK-OV-3 cell growth in a cell viability assay.
96
Total Activities
95
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SK-OV-3 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 96 | 5.51 | 8.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.82 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.58 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.43 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 8.20 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.08 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.41 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.30 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.00 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.85 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.75 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.65 |
| CHEMBL176544 | — | — | 1 | 6.40 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.34 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.33 |
| CHEMBL217354 | — | — | 1 | 6.28 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.28 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.17 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 6.15 |
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 5.97 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 2 | 5.92 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 5.91 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.81 |
| CHEMBL591429 | PAC-1 | 1.0 | 1 | 5.78 |
| CHEMBL585951 | — | — | 1 | 5.68 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 5.60 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 5.60 |
| CHEMBL1090090 | VX-702 | 2.0 | 1 | 5.58 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 5.39 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 5.35 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 5.35 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 1.495 | nM | 8.82 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 2.638 | nM | 8.58 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 3.751 | nM | 8.43 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 6.302 | nM | 8.20 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 8.386 | nM | 8.08 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 38.74 | nM | 7.41 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 50.12 | nM | 7.30 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 100.07 | nM | 7.00 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 142.64 | nM | 6.85 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 175.71 | nM | 6.75 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 224.36 | nM | 6.65 |
| CHEMBL176544 | — | IC50 | = | 396.65 | nM | 6.40 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 453.46 | nM | 6.34 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 467.59 | nM | 6.33 |
| CHEMBL217354 | — | IC50 | = | 527.13 | nM | 6.28 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 524.34 | nM | 6.28 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 671.87 | nM | 6.17 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 712.64 | nM | 6.15 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 1066.33 | nM | 5.97 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 1204.44 | nM | 5.92 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1220.89 | nM | 5.91 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1560.3 | nM | 5.81 |
| CHEMBL591429 | PAC-1 | IC50 | = | 1662.27 | nM | 5.78 |
| CHEMBL585951 | — | IC50 | = | 2070.97 | nM | 5.68 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 2490.65 | nM | 5.60 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 2502.49 | nM | 5.60 |
| CHEMBL1090090 | VX-702 | IC50 | = | 2616.97 | nM | 5.58 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 4062.26 | nM | 5.39 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 4481.49 | nM | 5.35 |
| CHEMBL939 | GEFITINIB | IC50 | = | 4460.42 | nM | 5.35 |
| CHEMBL379975 | — | IC50 | = | 4584.78 | nM | 5.34 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 4671.32 | nM | 5.33 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 4884.26 | nM | 5.31 |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 4993.4 | nM | 5.30 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 5718.1 | nM | 5.24 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 5911.21 | nM | 5.23 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 5998.16 | nM | 5.22 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 7210.91 | nM | 5.14 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 7394.32 | nM | 5.13 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 8155.03 | nM | 5.09 |
| CHEMBL191384 | — | IC50 | = | 8272.28 | nM | 5.08 |
| CHEMBL577784 | BX-795 | IC50 | = | 8278.2 | nM | 5.08 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 8467.65 | nM | 5.07 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 8713.29 | nM | 5.06 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 8797.72 | nM | 5.06 |
| CHEMBL1190711 | — | IC50 | = | 8831.93 | nM | 5.05 |
| CHEMBL2363137 | — | IC50 | = | 9127.05 | nM | 5.04 |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 9012.36 | nM | 5.04 |
| CHEMBL102714 | SB-216763 | IC50 | = | 9100.2 | nM | 5.04 |
| CHEMBL202721 | — | IC50 | = | 10552.2 | nM | 4.98 |