Assay Detail
Functional
CHEMBL2363668
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SANGER: Inhibition of human SNU-449 cell growth in a cell viability assay.
98
Total Activities
97
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SNU-449 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 98 | 5.46 | 8.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.72 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.38 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.86 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.85 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.69 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.12 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 6.89 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.88 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.84 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 6.76 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 6.71 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.68 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.52 |
| CHEMBL217354 | — | — | 1 | 6.43 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 6.41 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.31 |
| CHEMBL585951 | — | — | 1 | 6.28 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.26 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.24 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 6.21 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 6.14 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.09 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 6.08 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.02 |
| CHEMBL259181 | — | — | 1 | 5.96 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 5.91 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 5.70 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 5.59 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 5.59 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 5.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 1.905 | nM | 8.72 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 4.178 | nM | 8.38 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 13.77 | nM | 7.86 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 14.19 | nM | 7.85 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 20.26 | nM | 7.69 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 75.79 | nM | 7.12 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 127.72 | nM | 6.89 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 131.7 | nM | 6.88 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 142.75 | nM | 6.84 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 173.8 | nM | 6.76 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 194.29 | nM | 6.71 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 207.97 | nM | 6.68 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 299.64 | nM | 6.52 |
| CHEMBL217354 | — | IC50 | = | 372.39 | nM | 6.43 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 388.51 | nM | 6.41 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 492.52 | nM | 6.31 |
| CHEMBL585951 | — | IC50 | = | 522.47 | nM | 6.28 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 548.01 | nM | 6.26 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 575.19 | nM | 6.24 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 622.94 | nM | 6.21 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 727.48 | nM | 6.14 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 813.25 | nM | 6.09 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 827.35 | nM | 6.08 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 959.24 | nM | 6.02 |
| CHEMBL259181 | — | IC50 | = | 1092.79 | nM | 5.96 |
| CHEMBL939 | GEFITINIB | IC50 | = | 1222.08 | nM | 5.91 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1993.72 | nM | 5.70 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 2570.14 | nM | 5.59 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 2554.0 | nM | 5.59 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 2891.82 | nM | 5.54 |
| CHEMBL591429 | PAC-1 | IC50 | = | 3285.79 | nM | 5.48 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 3362.09 | nM | 5.47 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 3658.26 | nM | 5.44 |
| CHEMBL3349342 | — | IC50 | = | 3845.54 | nM | 5.42 |
| CHEMBL191384 | — | IC50 | = | 4866.49 | nM | 5.31 |
| CHEMBL577784 | BX-795 | IC50 | = | 4996.99 | nM | 5.30 |
| CHEMBL803 | CYTARABINE | IC50 | = | 5308.65 | nM | 5.28 |
| CHEMBL2363137 | — | IC50 | = | 5942.74 | nM | 5.23 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 6995.91 | nM | 5.16 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 7010.72 | nM | 5.15 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 7376.51 | nM | 5.13 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 7846.54 | nM | 5.11 |
| CHEMBL188678 | — | IC50 | = | 8279.3 | nM | 5.08 |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 8282.72 | nM | 5.08 |
| CHEMBL573107 | — | IC50 | = | 8752.65 | nM | 5.06 |
| CHEMBL1190711 | — | IC50 | = | 10847.43 | nM | 4.96 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 11607.18 | nM | 4.93 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 12212.7 | nM | 4.91 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 15043.51 | nM | 4.82 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 16420.44 | nM | 4.79 |