Assay Detail
Functional
CHEMBL2363673
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SANGER: Inhibition of human ST486 cell growth in a cell viability assay.
78
Total Activities
77
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | ST486 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 78 | 5.83 | 9.14 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.14 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.75 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.53 |
| CHEMBL9470 | SHIKONIN | — | 1 | 8.21 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 8.08 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 8.03 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.92 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.81 |
| CHEMBL514499 | GW843682X | — | 1 | 7.69 |
| CHEMBL300389 | — | — | 1 | 7.51 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.48 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.26 |
| CHEMBL1256459 | TORIN1 | — | 1 | 6.97 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 6.94 |
| CHEMBL512504 | — | — | 1 | 6.87 |
| CHEMBL585951 | — | — | 1 | 6.72 |
| CHEMBL379300 | A-443654 | — | 1 | 6.69 |
| CHEMBL572878 | TOZASERTIB | 2.0 | 1 | 6.64 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 6.53 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.46 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.31 |
| CHEMBL1190711 | — | — | 1 | 6.24 |
| CHEMBL941 | IMATINIB | 4.0 | 1 | 6.16 |
| CHEMBL27759 | ENTINOSTAT | 3.0 | 1 | 6.06 |
| CHEMBL591429 | PAC-1 | 1.0 | 1 | 6.01 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 5.90 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 5.89 |
| CHEMBL2144069 | — | — | 1 | 5.86 |
| CHEMBL217092 | SARACATINIB | 3.0 | 1 | 5.84 |
| CHEMBL1084546 | PF-00562271 | 1.0 | 1 | 5.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.7212 | nM | 9.14 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 1.767 | nM | 8.75 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 2.957 | nM | 8.53 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 6.179 | nM | 8.21 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 8.246 | nM | 8.08 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 9.406 | nM | 8.03 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 12.04 | nM | 7.92 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 15.53 | nM | 7.81 |
| CHEMBL514499 | GW843682X | IC50 | = | 20.36 | nM | 7.69 |
| CHEMBL300389 | — | IC50 | = | 31.22 | nM | 7.51 |
| CHEMBL513909 | BI-2536 | IC50 | = | 33.37 | nM | 7.48 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 55.25 | nM | 7.26 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 106.06 | nM | 6.97 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 114.06 | nM | 6.94 |
| CHEMBL512504 | — | IC50 | = | 135.27 | nM | 6.87 |
| CHEMBL585951 | — | IC50 | = | 189.67 | nM | 6.72 |
| CHEMBL379300 | A-443654 | IC50 | = | 203.93 | nM | 6.69 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 230.87 | nM | 6.64 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 296.14 | nM | 6.53 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 349.39 | nM | 6.46 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 494.36 | nM | 6.31 |
| CHEMBL1190711 | — | IC50 | = | 576.18 | nM | 6.24 |
| CHEMBL941 | IMATINIB | IC50 | = | 685.4 | nM | 6.16 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 879.17 | nM | 6.06 |
| CHEMBL591429 | PAC-1 | IC50 | = | 966.77 | nM | 6.01 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 1257.37 | nM | 5.90 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1281.17 | nM | 5.89 |
| CHEMBL2144069 | — | IC50 | = | 1386.62 | nM | 5.86 |
| CHEMBL217092 | SARACATINIB | IC50 | = | 1458.52 | nM | 5.84 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 1532.78 | nM | 5.82 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 1628.59 | nM | 5.79 |
| CHEMBL191384 | — | IC50 | = | 1742.33 | nM | 5.76 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 2085.18 | nM | 5.68 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 2249.88 | nM | 5.65 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 2410.48 | nM | 5.62 |
| CHEMBL601719 | CRIZOTINIB | IC50 | = | 2430.73 | nM | 5.61 |
| CHEMBL1673039 | — | IC50 | = | 3494.04 | nM | 5.46 |
| CHEMBL509032 | TAE-684 | IC50 | = | 3538.83 | nM | 5.45 |
| CHEMBL1336 | SORAFENIB | IC50 | = | 3836.73 | nM | 5.42 |
| CHEMBL2363137 | — | IC50 | = | 4829.21 | nM | 5.32 |
| CHEMBL472940 | — | IC50 | = | 4865.4 | nM | 5.31 |
| CHEMBL535 | SUNITINIB | IC50 | = | 6347.1 | nM | 5.20 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 6394.05 | nM | 5.19 |
| CHEMBL197603 | — | IC50 | = | 6439.69 | nM | 5.19 |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 8153.08 | nM | 5.09 |
| CHEMBL213100 | — | IC50 | = | 8272.27 | nM | 5.08 |
| CHEMBL221137 | EMBELIN | IC50 | = | 8301.83 | nM | 5.08 |
| CHEMBL180127 | SALUBRINAL | IC50 | = | 8536.8 | nM | 5.07 |
| CHEMBL36 | PYRIMETHAMINE | IC50 | = | 9308.24 | nM | 5.03 |
| CHEMBL401930 | — | IC50 | = | 9277.33 | nM | 5.03 |