Assay Detail
Functional
CHEMBL2363683
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SANGER: Inhibition of human SW1783 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SW1783 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.68 | 10.47 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 10.47 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.83 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.24 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 8.23 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.04 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.61 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.41 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.07 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.01 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 6.96 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 6.86 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.77 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.71 |
| CHEMBL217354 | — | — | 1 | 6.67 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 6.60 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 2 | 6.51 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.47 |
| CHEMBL585951 | — | — | 1 | 6.37 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 6.31 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.31 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.13 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.03 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.97 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 5.90 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 5.80 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 5.64 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 5.61 |
| CHEMBL135561 | — | — | 1 | 5.55 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 5.51 |
| CHEMBL577784 | BX-795 | — | 1 | 5.45 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | IC50 | = | 0.03355 | nM | 10.47 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 1.484 | nM | 8.83 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 5.7 | nM | 8.24 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 5.906 | nM | 8.23 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 9.236 | nM | 8.04 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 24.57 | nM | 7.61 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 38.58 | nM | 7.41 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 85.55 | nM | 7.07 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 97.99 | nM | 7.01 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 110.22 | nM | 6.96 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 139.04 | nM | 6.86 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 170.08 | nM | 6.77 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 193.05 | nM | 6.71 |
| CHEMBL217354 | — | IC50 | = | 213.01 | nM | 6.67 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 249.25 | nM | 6.60 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 305.83 | nM | 6.51 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 339.97 | nM | 6.47 |
| CHEMBL585951 | — | IC50 | = | 427.63 | nM | 6.37 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 487.45 | nM | 6.31 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 492.39 | nM | 6.31 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 733.37 | nM | 6.13 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 932.51 | nM | 6.03 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1068.84 | nM | 5.97 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 1260.3 | nM | 5.90 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 1600.84 | nM | 5.80 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 2310.7 | nM | 5.64 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 2470.78 | nM | 5.61 |
| CHEMBL135561 | — | IC50 | = | 2845.14 | nM | 5.55 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 3058.71 | nM | 5.51 |
| CHEMBL577784 | BX-795 | IC50 | = | 3543.76 | nM | 5.45 |
| CHEMBL803 | CYTARABINE | IC50 | = | 4613.83 | nM | 5.34 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 4753.08 | nM | 5.32 |
| CHEMBL191384 | — | IC50 | = | 6169.29 | nM | 5.21 |
| CHEMBL2363137 | — | IC50 | = | 7145.58 | nM | 5.15 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 7431.75 | nM | 5.13 |
| CHEMBL379975 | — | IC50 | = | 8481.07 | nM | 5.07 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 8573.47 | nM | 5.07 |
| CHEMBL221137 | EMBELIN | IC50 | = | 10066.15 | nM | 5.00 |
| CHEMBL591429 | PAC-1 | IC50 | = | 11012.06 | nM | 4.96 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 10996.27 | nM | 4.96 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 14239.12 | nM | 4.85 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 15764.74 | nM | 4.80 |
| CHEMBL188678 | — | IC50 | = | 16099.32 | nM | 4.79 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 17128.01 | nM | 4.77 |
| CHEMBL573107 | — | IC50 | = | 16999.77 | nM | 4.77 |
| CHEMBL939 | GEFITINIB | IC50 | = | 17641.45 | nM | 4.75 |
| CHEMBL3349342 | — | IC50 | = | 19718.51 | nM | 4.71 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 19577.48 | nM | 4.71 |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 19780.65 | nM | 4.70 |
| CHEMBL258844 | — | IC50 | = | 22374.41 | nM | 4.65 |