Assay Detail
Functional
CHEMBL2363712
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SANGER: Inhibition of human 647-V cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | 647-V |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.52 | 9.61 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 9.61 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.05 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.73 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.62 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.16 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.86 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.73 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.68 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.64 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.11 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.06 |
| CHEMBL217354 | — | — | 1 | 7.05 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.98 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 6.83 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.48 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.45 |
| CHEMBL585951 | — | — | 1 | 6.40 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.34 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.31 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.21 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.17 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.00 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.00 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 5.91 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 5.81 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 5.76 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 5.64 |
| CHEMBL2363137 | — | — | 1 | 5.51 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 5.50 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 5.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | IC50 | = | 0.2481 | nM | 9.61 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.8964 | nM | 9.05 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.842 | nM | 8.73 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 2.416 | nM | 8.62 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 6.905 | nM | 8.16 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 13.71 | nM | 7.86 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 18.81 | nM | 7.73 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 20.89 | nM | 7.68 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 23.03 | nM | 7.64 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 78.07 | nM | 7.11 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 87.39 | nM | 7.06 |
| CHEMBL217354 | — | IC50 | = | 88.43 | nM | 7.05 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 104.08 | nM | 6.98 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 149.42 | nM | 6.83 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 331.89 | nM | 6.48 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 358.52 | nM | 6.45 |
| CHEMBL585951 | — | IC50 | = | 401.43 | nM | 6.40 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 455.41 | nM | 6.34 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 487.34 | nM | 6.31 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 617.87 | nM | 6.21 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 681.48 | nM | 6.17 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 1006.95 | nM | 6.00 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 1000.03 | nM | 6.00 |
| CHEMBL803 | CYTARABINE | IC50 | = | 1232.74 | nM | 5.91 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 1538.8 | nM | 5.81 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 1733.41 | nM | 5.76 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 2304.55 | nM | 5.64 |
| CHEMBL2363137 | — | IC50 | = | 3086.93 | nM | 5.51 |
| CHEMBL939 | GEFITINIB | IC50 | = | 3162.2 | nM | 5.50 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 3984.52 | nM | 5.40 |
| CHEMBL379975 | — | IC50 | = | 4104.07 | nM | 5.39 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 4440.22 | nM | 5.35 |
| CHEMBL135561 | — | IC50 | = | 4710.15 | nM | 5.33 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 5620.42 | nM | 5.25 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 5747.06 | nM | 5.24 |
| CHEMBL258844 | — | IC50 | = | 5877.3 | nM | 5.23 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 5991.48 | nM | 5.22 |
| CHEMBL1190711 | — | IC50 | = | 7297.41 | nM | 5.14 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 9307.22 | nM | 5.03 |
| CHEMBL573107 | — | IC50 | = | 11597.41 | nM | 4.94 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 12005.81 | nM | 4.92 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 12097.24 | nM | 4.92 |
| CHEMBL2134202 | — | IC50 | = | 12358.21 | nM | 4.91 |
| CHEMBL1186585 | — | IC50 | = | 14732.56 | nM | 4.83 |
| CHEMBL188678 | — | IC50 | = | 15270.53 | nM | 4.82 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 15927.02 | nM | 4.80 |
| CHEMBL591429 | PAC-1 | IC50 | = | 17294.82 | nM | 4.76 |
| CHEMBL259181 | — | IC50 | = | 19351.54 | nM | 4.71 |
| CHEMBL221137 | EMBELIN | IC50 | = | 24543.03 | nM | 4.61 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 26881.09 | nM | 4.57 |