Assay Detail
Functional
CHEMBL2363747
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SANGER: Inhibition of human BB30-HNC cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | BB30-HNC |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.88 | 9.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.70 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 9.64 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 9.47 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 9.40 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 9.01 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.98 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 8.50 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.08 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 8.07 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 8.02 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 7.79 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.67 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.53 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.51 |
| CHEMBL514499 | GW843682X | — | 1 | 7.47 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.45 |
| CHEMBL300389 | — | — | 1 | 7.28 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 7.26 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.24 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.19 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 7.19 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 7.07 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 7.03 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.96 |
| CHEMBL585951 | — | — | 1 | 6.91 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 6.88 |
| CHEMBL553 | ERLOTINIB | 4.0 | 1 | 6.83 |
| CHEMBL217354 | — | — | 1 | 6.79 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 6.78 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.76 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.2008 | nM | 9.70 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 0.2312 | nM | 9.64 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 0.3353 | nM | 9.47 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 0.3988 | nM | 9.40 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 0.9842 | nM | 9.01 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.049 | nM | 8.98 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 3.138 | nM | 8.50 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 8.315 | nM | 8.08 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 8.578 | nM | 8.07 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 9.521 | nM | 8.02 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 16.34 | nM | 7.79 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 21.55 | nM | 7.67 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 29.85 | nM | 7.53 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 30.61 | nM | 7.51 |
| CHEMBL514499 | GW843682X | IC50 | = | 34.15 | nM | 7.47 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 35.35 | nM | 7.45 |
| CHEMBL300389 | — | IC50 | = | 52.49 | nM | 7.28 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 54.37 | nM | 7.26 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 57.3 | nM | 7.24 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 64.18 | nM | 7.19 |
| CHEMBL513909 | BI-2536 | IC50 | = | 64.36 | nM | 7.19 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 85.51 | nM | 7.07 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 94.28 | nM | 7.03 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 110.15 | nM | 6.96 |
| CHEMBL585951 | — | IC50 | = | 122.37 | nM | 6.91 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 130.78 | nM | 6.88 |
| CHEMBL553 | ERLOTINIB | IC50 | = | 147.65 | nM | 6.83 |
| CHEMBL217354 | — | IC50 | = | 161.74 | nM | 6.79 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 165.76 | nM | 6.78 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 173.3 | nM | 6.76 |
| CHEMBL379300 | A-443654 | IC50 | = | 219.63 | nM | 6.66 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 225.91 | nM | 6.65 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 243.49 | nM | 6.61 |
| CHEMBL554 | LAPATINIB | IC50 | = | 246.54 | nM | 6.61 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 315.25 | nM | 6.50 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 323.67 | nM | 6.49 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 388.32 | nM | 6.41 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 585.23 | nM | 6.23 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 663.81 | nM | 6.18 |
| CHEMBL197603 | — | IC50 | = | 873.83 | nM | 6.06 |
| CHEMBL217092 | SARACATINIB | IC50 | = | 862.03 | nM | 6.06 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 924.69 | nM | 6.03 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 935.31 | nM | 6.03 |
| CHEMBL509032 | TAE-684 | IC50 | = | 1131.12 | nM | 5.95 |
| CHEMBL401930 | — | IC50 | = | 1124.18 | nM | 5.95 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 1188.51 | nM | 5.92 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 1287.14 | nM | 5.89 |
| CHEMBL379975 | — | IC50 | = | 1357.67 | nM | 5.87 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 1389.78 | nM | 5.86 |
| CHEMBL3349342 | — | IC50 | = | 1581.4 | nM | 5.80 |