Assay Detail
Functional
CHEMBL2363752
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SANGER: Inhibition of human BCPAP cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | BCPAP |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.87 | 9.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 9.35 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.24 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.02 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.87 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 8.84 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.63 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.53 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.52 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.73 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.58 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 7.37 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.28 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.23 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.23 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.99 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.87 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.72 |
| CHEMBL217354 | — | — | 1 | 6.62 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.62 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.53 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.44 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 6.30 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.30 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.23 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.13 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 6.06 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.04 |
| CHEMBL585951 | — | — | 1 | 6.03 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.01 |
| CHEMBL1084546 | PF-00562271 | 1.0 | 1 | 5.99 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 0.448 | nM | 9.35 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.5813 | nM | 9.24 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 0.9466 | nM | 9.02 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 1.345 | nM | 8.87 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 1.452 | nM | 8.84 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 2.33 | nM | 8.63 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 2.978 | nM | 8.53 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 3.041 | nM | 8.52 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 18.65 | nM | 7.73 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 26.46 | nM | 7.58 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 43.1 | nM | 7.37 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 52.5 | nM | 7.28 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 58.53 | nM | 7.23 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 58.92 | nM | 7.23 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 101.62 | nM | 6.99 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 135.25 | nM | 6.87 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 188.72 | nM | 6.72 |
| CHEMBL217354 | — | IC50 | = | 241.64 | nM | 6.62 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 239.6 | nM | 6.62 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 298.79 | nM | 6.53 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 360.01 | nM | 6.44 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 501.42 | nM | 6.30 |
| CHEMBL803 | CYTARABINE | IC50 | = | 501.18 | nM | 6.30 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 587.91 | nM | 6.23 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 736.95 | nM | 6.13 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 877.37 | nM | 6.06 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 922.59 | nM | 6.04 |
| CHEMBL585951 | — | IC50 | = | 932.35 | nM | 6.03 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 969.6 | nM | 6.01 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 1012.88 | nM | 5.99 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 1317.07 | nM | 5.88 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 1435.14 | nM | 5.84 |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 1668.98 | nM | 5.78 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 1664.57 | nM | 5.78 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 1886.76 | nM | 5.72 |
| CHEMBL2363137 | — | IC50 | = | 2049.79 | nM | 5.69 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 2127.4 | nM | 5.67 |
| CHEMBL3349342 | — | IC50 | = | 2180.49 | nM | 5.66 |
| CHEMBL577784 | BX-795 | IC50 | = | 2231.58 | nM | 5.65 |
| CHEMBL939 | GEFITINIB | IC50 | = | 3082.95 | nM | 5.51 |
| CHEMBL1190711 | — | IC50 | = | 3172.78 | nM | 5.50 |
| CHEMBL191384 | — | IC50 | = | 4451.48 | nM | 5.35 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 4634.81 | nM | 5.33 |
| CHEMBL105442 | CI-1040 | IC50 | = | 5329.69 | nM | 5.27 |
| CHEMBL1230020 | PLX-4720 | IC50 | = | 7217.64 | nM | 5.14 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 8277.52 | nM | 5.08 |
| CHEMBL255863 | NILOTINIB | IC50 | = | 9025.62 | nM | 5.04 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 12474.93 | nM | 4.90 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 13044.41 | nM | 4.88 |
| CHEMBL591429 | PAC-1 | IC50 | = | 13582.8 | nM | 4.87 |