Assay Detail
Functional
CHEMBL2363758
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SANGER: Inhibition of human BHY cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | BHY |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.76 | 9.71 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.71 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 9.22 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 8.94 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.67 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.65 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.28 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.00 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.81 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.72 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.54 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.37 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.12 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 6.97 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.62 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.61 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 6.54 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.53 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.44 |
| CHEMBL585951 | — | — | 1 | 6.29 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.25 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.16 |
| CHEMBL217354 | — | — | 1 | 6.15 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.06 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.05 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.05 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 6.01 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 5.98 |
| CHEMBL379975 | — | — | 1 | 5.94 |
| CHEMBL288441 | BOSUTINIB | 4.0 | 1 | 5.91 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 5.86 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.1954 | nM | 9.71 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 0.6007 | nM | 9.22 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 1.141 | nM | 8.94 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 2.16 | nM | 8.67 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 2.258 | nM | 8.65 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 5.31 | nM | 8.28 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 9.946 | nM | 8.00 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 15.33 | nM | 7.81 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 19.12 | nM | 7.72 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 28.88 | nM | 7.54 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 42.72 | nM | 7.37 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 75.28 | nM | 7.12 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 107.06 | nM | 6.97 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 236.91 | nM | 6.62 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 245.55 | nM | 6.61 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 286.55 | nM | 6.54 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 297.13 | nM | 6.53 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 364.8 | nM | 6.44 |
| CHEMBL585951 | — | IC50 | = | 510.17 | nM | 6.29 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 563.96 | nM | 6.25 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 688.04 | nM | 6.16 |
| CHEMBL217354 | — | IC50 | = | 701.65 | nM | 6.15 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 872.49 | nM | 6.06 |
| CHEMBL803 | CYTARABINE | IC50 | = | 897.62 | nM | 6.05 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 887.34 | nM | 6.05 |
| CHEMBL939 | GEFITINIB | IC50 | = | 975.48 | nM | 6.01 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 1045.79 | nM | 5.98 |
| CHEMBL379975 | — | IC50 | = | 1150.14 | nM | 5.94 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 1228.92 | nM | 5.91 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1374.13 | nM | 5.86 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 1469.23 | nM | 5.83 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 1531.69 | nM | 5.82 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 1656.63 | nM | 5.78 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 1827.47 | nM | 5.74 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 1810.34 | nM | 5.74 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 2349.12 | nM | 5.63 |
| CHEMBL1190711 | — | IC50 | = | 2814.27 | nM | 5.55 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 3255.71 | nM | 5.49 |
| CHEMBL3349342 | — | IC50 | = | 3285.08 | nM | 5.48 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 4124.95 | nM | 5.38 |
| CHEMBL2363137 | — | IC50 | = | 4498.78 | nM | 5.35 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 4918.97 | nM | 5.31 |
| CHEMBL259181 | — | IC50 | = | 5131.58 | nM | 5.29 |
| CHEMBL573107 | — | IC50 | = | 5510.7 | nM | 5.26 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 5725.8 | nM | 5.24 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 6000.34 | nM | 5.22 |
| CHEMBL221137 | EMBELIN | IC50 | = | 6032.66 | nM | 5.22 |
| CHEMBL577784 | BX-795 | IC50 | = | 7681.98 | nM | 5.12 |
| CHEMBL135561 | — | IC50 | = | 7988.6 | nM | 5.10 |
| CHEMBL191384 | — | IC50 | = | 8672.38 | nM | 5.06 |