Assay Detail
Functional
CHEMBL2363762
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SANGER: Inhibition of human BPH-1 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | BPH-1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.89 | 9.28 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.28 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 9.22 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.99 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.72 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.68 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.49 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 8.40 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 8.32 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 8.22 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.99 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.69 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.66 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.52 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.49 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 7.23 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 7.22 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.08 |
| CHEMBL3349342 | — | — | 1 | 6.87 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.87 |
| CHEMBL1614701 | SELUMETINIB | 4.0 | 1 | 6.74 |
| CHEMBL217354 | — | — | 1 | 6.54 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 6.50 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 6.31 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.25 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 6.11 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.05 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.03 |
| CHEMBL379975 | — | — | 1 | 5.97 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.90 |
| CHEMBL1084546 | PF-00562271 | 1.0 | 1 | 5.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.5205 | nM | 9.28 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 0.5996 | nM | 9.22 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.022 | nM | 8.99 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 1.899 | nM | 8.72 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 2.082 | nM | 8.68 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 3.263 | nM | 8.49 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 3.95 | nM | 8.40 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 4.756 | nM | 8.32 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 6.027 | nM | 8.22 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 10.3 | nM | 7.99 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 20.28 | nM | 7.69 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 22.12 | nM | 7.66 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 29.9 | nM | 7.52 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 32.39 | nM | 7.49 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 59.09 | nM | 7.23 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 59.88 | nM | 7.22 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 83.14 | nM | 7.08 |
| CHEMBL3349342 | — | IC50 | = | 134.79 | nM | 6.87 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 134.1 | nM | 6.87 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 182.31 | nM | 6.74 |
| CHEMBL217354 | — | IC50 | = | 285.81 | nM | 6.54 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 314.0 | nM | 6.50 |
| CHEMBL939 | GEFITINIB | IC50 | = | 491.16 | nM | 6.31 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 563.44 | nM | 6.25 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 772.41 | nM | 6.11 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 883.95 | nM | 6.05 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 942.82 | nM | 6.03 |
| CHEMBL379975 | — | IC50 | = | 1066.51 | nM | 5.97 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1259.99 | nM | 5.90 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 1287.66 | nM | 5.89 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 1304.75 | nM | 5.88 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 1448.05 | nM | 5.84 |
| CHEMBL105442 | CI-1040 | IC50 | = | 1895.91 | nM | 5.72 |
| CHEMBL585951 | — | IC50 | = | 1973.49 | nM | 5.71 |
| CHEMBL1190711 | — | IC50 | = | 1990.92 | nM | 5.70 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 2070.98 | nM | 5.68 |
| CHEMBL573107 | — | IC50 | = | 2129.57 | nM | 5.67 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 2244.9 | nM | 5.65 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 2658.5 | nM | 5.58 |
| CHEMBL393929 | — | IC50 | = | 2974.55 | nM | 5.53 |
| CHEMBL577784 | BX-795 | IC50 | = | 3135.23 | nM | 5.50 |
| CHEMBL803 | CYTARABINE | IC50 | = | 3642.05 | nM | 5.44 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 3819.9 | nM | 5.42 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 4298.47 | nM | 5.37 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 4900.33 | nM | 5.31 |
| CHEMBL135561 | — | IC50 | = | 6321.41 | nM | 5.20 |
| CHEMBL202721 | — | IC50 | = | 6500.75 | nM | 5.19 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 6802.76 | nM | 5.17 |
| CHEMBL38 | TRETINOIN | IC50 | = | 7436.11 | nM | 5.13 |
| CHEMBL1173055 | RUCAPARIB | IC50 | = | 8152.08 | nM | 5.09 |