Assay Detail
Functional
CHEMBL2363766
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SANGER: Inhibition of human BV-173 cell growth in a cell viability assay.
126
Total Activities
125
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | BV-173 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 126 | 5.98 | 9.29 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL213100 | — | — | 1 | 9.29 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.62 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.55 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.28 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.27 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 8.22 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 8.20 |
| CHEMBL255863 | NILOTINIB | 4.0 | 1 | 7.96 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.76 |
| CHEMBL514499 | GW843682X | — | 1 | 7.75 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.66 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 7.64 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.62 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.59 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.52 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.46 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.37 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.36 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 7.08 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 7.04 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 6.95 |
| CHEMBL1090090 | VX-702 | 2.0 | 1 | 6.94 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 6.91 |
| CHEMBL572878 | TOZASERTIB | 2.0 | 1 | 6.90 |
| CHEMBL300389 | — | — | 1 | 6.84 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 6.75 |
| CHEMBL941 | IMATINIB | 4.0 | 1 | 6.73 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 6.73 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 6.72 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL213100 | — | IC50 | = | 0.5143 | nM | 9.29 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 2.381 | nM | 8.62 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 2.807 | nM | 8.55 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 5.3 | nM | 8.28 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 5.387 | nM | 8.27 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 6.067 | nM | 8.22 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 6.349 | nM | 8.20 |
| CHEMBL255863 | NILOTINIB | IC50 | = | 10.89 | nM | 7.96 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 17.27 | nM | 7.76 |
| CHEMBL514499 | GW843682X | IC50 | = | 17.74 | nM | 7.75 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 22.03 | nM | 7.66 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 23.14 | nM | 7.64 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 23.87 | nM | 7.62 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 25.54 | nM | 7.59 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 30.41 | nM | 7.52 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 34.26 | nM | 7.46 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 42.27 | nM | 7.37 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 43.85 | nM | 7.36 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 83.97 | nM | 7.08 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 90.61 | nM | 7.04 |
| CHEMBL513909 | BI-2536 | IC50 | = | 112.43 | nM | 6.95 |
| CHEMBL1090090 | VX-702 | IC50 | = | 113.86 | nM | 6.94 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 122.71 | nM | 6.91 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 126.41 | nM | 6.90 |
| CHEMBL300389 | — | IC50 | = | 144.34 | nM | 6.84 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 175.96 | nM | 6.75 |
| CHEMBL939 | GEFITINIB | IC50 | = | 186.55 | nM | 6.73 |
| CHEMBL941 | IMATINIB | IC50 | = | 187.4 | nM | 6.73 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 190.2 | nM | 6.72 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 250.77 | nM | 6.60 |
| CHEMBL379300 | A-443654 | IC50 | = | 268.78 | nM | 6.57 |
| CHEMBL483847 | — | IC50 | = | 285.53 | nM | 6.54 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 345.96 | nM | 6.46 |
| CHEMBL197603 | — | IC50 | = | 345.47 | nM | 6.46 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 369.48 | nM | 6.43 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 371.21 | nM | 6.43 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 393.2 | nM | 6.41 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 435.95 | nM | 6.36 |
| CHEMBL379975 | — | IC50 | = | 434.2 | nM | 6.36 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 507.92 | nM | 6.29 |
| CHEMBL803 | CYTARABINE | IC50 | = | 515.51 | nM | 6.29 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 582.44 | nM | 6.24 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 652.48 | nM | 6.18 |
| CHEMBL217092 | SARACATINIB | IC50 | = | 652.49 | nM | 6.18 |
| CHEMBL2144069 | — | IC50 | = | 691.54 | nM | 6.16 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 686.79 | nM | 6.16 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 748.02 | nM | 6.13 |
| CHEMBL585951 | — | IC50 | = | 736.48 | nM | 6.13 |
| CHEMBL477989 | SB590885 | IC50 | = | 770.55 | nM | 6.11 |
| CHEMBL1230020 | PLX-4720 | IC50 | = | 796.44 | nM | 6.10 |