Assay Detail
Functional
CHEMBL2363832
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SANGER: Inhibition of human CAMA-1 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CAMA-1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.34 | 8.88 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.88 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 8.32 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 8.01 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.98 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 7.89 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.50 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.34 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.20 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.06 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.89 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.80 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.54 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 6.40 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 6.40 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.36 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.27 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.21 |
| CHEMBL217354 | — | — | 1 | 6.18 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 6.08 |
| CHEMBL2363137 | — | — | 1 | 6.04 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 5.98 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 2 | 5.92 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.82 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 5.76 |
| CHEMBL591429 | PAC-1 | 1.0 | 1 | 5.56 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 5.41 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 5.36 |
| CHEMBL221137 | EMBELIN | — | 1 | 5.15 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 5.07 |
| CHEMBL1023 | BEXAROTENE | 4.0 | 1 | 5.06 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.307 | nM | 8.88 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 4.771 | nM | 8.32 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 9.799 | nM | 8.01 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 10.45 | nM | 7.98 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 12.93 | nM | 7.89 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 32.01 | nM | 7.50 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 45.57 | nM | 7.34 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 63.03 | nM | 7.20 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 87.43 | nM | 7.06 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 129.24 | nM | 6.89 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 159.33 | nM | 6.80 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 289.13 | nM | 6.54 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 395.8 | nM | 6.40 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 394.59 | nM | 6.40 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 436.26 | nM | 6.36 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 540.59 | nM | 6.27 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 621.52 | nM | 6.21 |
| CHEMBL217354 | — | IC50 | = | 660.73 | nM | 6.18 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 833.94 | nM | 6.08 |
| CHEMBL2363137 | — | IC50 | = | 911.31 | nM | 6.04 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 1037.35 | nM | 5.98 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 1200.1 | nM | 5.92 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1516.69 | nM | 5.82 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 1719.71 | nM | 5.76 |
| CHEMBL591429 | PAC-1 | IC50 | = | 2751.38 | nM | 5.56 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 3937.34 | nM | 5.41 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 4352.0 | nM | 5.36 |
| CHEMBL221137 | EMBELIN | IC50 | = | 7091.9 | nM | 5.15 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 8521.62 | nM | 5.07 |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 8634.83 | nM | 5.06 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 8771.46 | nM | 5.06 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 9060.12 | nM | 5.04 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 9281.28 | nM | 5.03 |
| CHEMBL259181 | — | IC50 | = | 9647.86 | nM | 5.02 |
| CHEMBL939 | GEFITINIB | IC50 | = | 12163.26 | nM | 4.92 |
| CHEMBL409 | BICALUTAMIDE | IC50 | = | 12392.59 | nM | 4.91 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 13004.56 | nM | 4.89 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 17524.73 | nM | 4.76 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 18663.36 | nM | 4.73 |
| CHEMBL202721 | — | IC50 | = | 20881.01 | nM | 4.68 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 20980.3 | nM | 4.68 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 21295.8 | nM | 4.67 |
| CHEMBL477989 | SB590885 | IC50 | = | 23240.72 | nM | 4.63 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 24079.67 | nM | 4.62 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 25125.22 | nM | 4.60 |
| CHEMBL1090090 | VX-702 | IC50 | = | 25910.21 | nM | 4.59 |
| CHEMBL573107 | — | IC50 | = | 26487.58 | nM | 4.58 |
| CHEMBL577784 | BX-795 | IC50 | = | 27112.8 | nM | 4.57 |
| CHEMBL38 | TRETINOIN | IC50 | = | 28017.88 | nM | 4.55 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 27907.21 | nM | 4.55 |