Assay Detail
Functional
CHEMBL2363835
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SANGER: Inhibition of human CCF-STTG1 cell growth in a cell viability assay.
38
Total Activities
38
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CCF-STTG1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 38 | 5.85 | 8.53 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 8.53 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.23 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.08 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.50 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.45 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.17 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.67 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.65 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.60 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 6.29 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.26 |
| CHEMBL585951 | — | — | 1 | 6.21 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.12 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.03 |
| CHEMBL477772 | PAZOPANIB | 4.0 | 1 | 5.98 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 1 | 5.85 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 5.34 |
| CHEMBL409 | BICALUTAMIDE | 4.0 | 1 | 5.31 |
| CHEMBL191384 | — | — | 1 | 5.19 |
| CHEMBL512504 | — | — | 1 | 5.17 |
| CHEMBL258844 | — | — | 1 | 5.17 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 5.16 |
| CHEMBL1190711 | — | — | 1 | 5.14 |
| CHEMBL558642 | GSK-650394 | — | 1 | 4.90 |
| CHEMBL2363137 | — | — | 1 | 4.89 |
| CHEMBL1084546 | PF-00562271 | 1.0 | 1 | 4.87 |
| CHEMBL221137 | EMBELIN | — | 1 | 4.86 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 4.56 |
| CHEMBL1023 | BEXAROTENE | 4.0 | 1 | 4.37 |
| CHEMBL259181 | — | — | 1 | 4.34 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL252164 | LUMINESPIB | IC50 | = | 2.974 | nM | 8.53 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 5.826 | nM | 8.23 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 8.373 | nM | 8.08 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 31.42 | nM | 7.50 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 35.5 | nM | 7.45 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 67.29 | nM | 7.17 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 215.59 | nM | 6.67 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 224.75 | nM | 6.65 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 253.35 | nM | 6.60 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 513.74 | nM | 6.29 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 551.34 | nM | 6.26 |
| CHEMBL585951 | — | IC50 | = | 623.83 | nM | 6.21 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 768.01 | nM | 6.12 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 926.37 | nM | 6.03 |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 1049.81 | nM | 5.98 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 1425.25 | nM | 5.85 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 4562.09 | nM | 5.34 |
| CHEMBL409 | BICALUTAMIDE | IC50 | = | 4929.29 | nM | 5.31 |
| CHEMBL191384 | — | IC50 | = | 6407.06 | nM | 5.19 |
| CHEMBL512504 | — | IC50 | = | 6749.02 | nM | 5.17 |
| CHEMBL258844 | — | IC50 | = | 6815.01 | nM | 5.17 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 6911.49 | nM | 5.16 |
| CHEMBL1190711 | — | IC50 | = | 7239.49 | nM | 5.14 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 12599.69 | nM | 4.90 |
| CHEMBL2363137 | — | IC50 | = | 12750.54 | nM | 4.89 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 13403.86 | nM | 4.87 |
| CHEMBL221137 | EMBELIN | IC50 | = | 13953.41 | nM | 4.86 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 27812.48 | nM | 4.56 |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 42465.97 | nM | 4.37 |
| CHEMBL259181 | — | IC50 | = | 46159.23 | nM | 4.34 |
| CHEMBL135561 | — | IC50 | = | 69098.15 | nM | 4.16 |
| CHEMBL591429 | PAC-1 | IC50 | = | 82163.98 | nM | 4.08 |
| CHEMBL472940 | — | IC50 | = | 1255895.32 | nM | - |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 103342.22 | nM | - |
| CHEMBL228043 | — | IC50 | = | 941874.46 | nM | - |
| CHEMBL92309 | — | IC50 | = | 4014495.64 | nM | - |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 143334.49 | nM | - |
| CHEMBL472004 | — | IC50 | = | 126506.41 | nM | - |