Assay Detail
Functional
CHEMBL2363843
Review assay metadata, readout intent, target linkage, and publication context from the same page.
SANGER: Inhibition of human CHP-212 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHP-212 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 6.04 | 9.28 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 9.28 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.14 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.99 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 8.56 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.52 |
| CHEMBL1614701 | SELUMETINIB | 4.0 | 1 | 8.50 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.45 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 8.36 |
| CHEMBL3349342 | — | — | 1 | 8.31 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.23 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.13 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.66 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.61 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 7.58 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 7.54 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 7.47 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.46 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 7.32 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.28 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.12 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.09 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 7.08 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 7.06 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 6.83 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 6.82 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.70 |
| CHEMBL585951 | — | — | 1 | 6.54 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.36 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 6.34 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 6.23 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 0.5273 | nM | 9.28 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 0.7298 | nM | 9.14 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 1.026 | nM | 8.99 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 2.752 | nM | 8.56 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 3.001 | nM | 8.52 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 3.153 | nM | 8.50 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 3.547 | nM | 8.45 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 4.368 | nM | 8.36 |
| CHEMBL3349342 | — | IC50 | = | 4.918 | nM | 8.31 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 5.828 | nM | 8.23 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 7.342 | nM | 8.13 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 22.12 | nM | 7.66 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 24.59 | nM | 7.61 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 26.28 | nM | 7.58 |
| CHEMBL105442 | CI-1040 | IC50 | = | 28.85 | nM | 7.54 |
| CHEMBL803 | CYTARABINE | IC50 | = | 33.47 | nM | 7.47 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 34.96 | nM | 7.46 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 47.95 | nM | 7.32 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 52.43 | nM | 7.28 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 74.95 | nM | 7.12 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 80.95 | nM | 7.09 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 82.16 | nM | 7.08 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 87.73 | nM | 7.06 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 147.74 | nM | 6.83 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 151.62 | nM | 6.82 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 197.82 | nM | 6.70 |
| CHEMBL585951 | — | IC50 | = | 286.38 | nM | 6.54 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 436.97 | nM | 6.36 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 457.53 | nM | 6.34 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 593.59 | nM | 6.23 |
| CHEMBL379975 | — | IC50 | = | 619.0 | nM | 6.21 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1096.47 | nM | 5.96 |
| CHEMBL577784 | BX-795 | IC50 | = | 1140.37 | nM | 5.94 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 1378.65 | nM | 5.86 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 1410.96 | nM | 5.85 |
| CHEMBL202721 | — | IC50 | = | 1468.59 | nM | 5.83 |
| CHEMBL191334 | NUTLIN-3 | IC50 | = | 1813.69 | nM | 5.74 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 2095.39 | nM | 5.68 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 2184.42 | nM | 5.66 |
| CHEMBL2363137 | — | IC50 | = | 2576.97 | nM | 5.59 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 2820.91 | nM | 5.55 |
| CHEMBL221137 | EMBELIN | IC50 | = | 3121.54 | nM | 5.51 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 3925.49 | nM | 5.41 |
| CHEMBL217354 | — | IC50 | = | 4572.37 | nM | 5.34 |
| CHEMBL258844 | — | IC50 | = | 4558.67 | nM | 5.34 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 5394.09 | nM | 5.27 |
| CHEMBL1190711 | — | IC50 | = | 6453.24 | nM | 5.19 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 6482.67 | nM | 5.19 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 7518.96 | nM | 5.12 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 7847.41 | nM | 5.11 |