Assay Detail
Functional
CHEMBL2363845
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SANGER: Inhibition of human COLO-205 cell growth in a cell viability assay.
38
Total Activities
38
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | COLO-205 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 38 | 6.15 | 9.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.10 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.86 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 8.65 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.50 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.84 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.57 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.31 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.24 |
| CHEMBL1091644 | LINSITINIB | 3.0 | 1 | 6.98 |
| CHEMBL585951 | — | — | 1 | 6.82 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.79 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.58 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.36 |
| CHEMBL1084546 | PF-00562271 | 1.0 | 1 | 6.31 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.27 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 5.83 |
| CHEMBL258844 | — | — | 1 | 5.70 |
| CHEMBL259181 | — | — | 1 | 5.64 |
| CHEMBL1190711 | — | — | 1 | 5.63 |
| CHEMBL2363137 | — | — | 1 | 5.59 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 5.49 |
| CHEMBL221137 | EMBELIN | — | 1 | 5.41 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 5.38 |
| CHEMBL412142 | LADUVIGLUSIB | 1.0 | 1 | 5.03 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 1 | 4.71 |
| CHEMBL191384 | — | — | 1 | 4.68 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 4.53 |
| CHEMBL591429 | PAC-1 | 1.0 | 1 | 4.52 |
| CHEMBL135561 | — | — | 1 | 4.47 |
| CHEMBL512504 | — | — | 1 | 4.43 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.8015 | nM | 9.10 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 1.368 | nM | 8.86 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 2.243 | nM | 8.65 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 3.153 | nM | 8.50 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 14.33 | nM | 7.84 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 26.99 | nM | 7.57 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 49.19 | nM | 7.31 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 57.16 | nM | 7.24 |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 104.54 | nM | 6.98 |
| CHEMBL585951 | — | IC50 | = | 151.54 | nM | 6.82 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 162.42 | nM | 6.79 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 264.97 | nM | 6.58 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 432.22 | nM | 6.36 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 486.58 | nM | 6.31 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 537.72 | nM | 6.27 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 1471.81 | nM | 5.83 |
| CHEMBL258844 | — | IC50 | = | 1997.06 | nM | 5.70 |
| CHEMBL259181 | — | IC50 | = | 2293.82 | nM | 5.64 |
| CHEMBL1190711 | — | IC50 | = | 2350.82 | nM | 5.63 |
| CHEMBL2363137 | — | IC50 | = | 2549.22 | nM | 5.59 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 3244.54 | nM | 5.49 |
| CHEMBL221137 | EMBELIN | IC50 | = | 3867.4 | nM | 5.41 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 4178.64 | nM | 5.38 |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 9438.21 | nM | 5.03 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 19311.1 | nM | 4.71 |
| CHEMBL191384 | — | IC50 | = | 21102.55 | nM | 4.68 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 29394.42 | nM | 4.53 |
| CHEMBL591429 | PAC-1 | IC50 | = | 30244.49 | nM | 4.52 |
| CHEMBL135561 | — | IC50 | = | 34231.01 | nM | 4.47 |
| CHEMBL512504 | — | IC50 | = | 37258.87 | nM | 4.43 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 38441.75 | nM | 4.42 |
| CHEMBL409 | BICALUTAMIDE | IC50 | = | 66326.93 | nM | 4.18 |
| CHEMBL472940 | — | IC50 | = | 1369913.67 | nM | - |
| CHEMBL92309 | — | IC50 | = | 9809788.57 | nM | - |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 173940.97 | nM | - |
| CHEMBL228043 | — | IC50 | = | 105058.67 | nM | - |
| CHEMBL472004 | — | IC50 | = | 962301.68 | nM | - |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 493503.03 | nM | - |