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Assay Detail

CHEMBL2380041

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Binding
Inhibition of muscarinic acetylcholine receptor in rat cortex
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Discovery of subtype selective muscarinic receptor antagonists as alternatives to atropine using in silico pharmacophore modeling and virtual screening methods.
Bhattacharjee AK, Pomponio JW, Evans SA, Pervitsky D, Gordon RK.
Bioorg Med Chem (2013) 21 : 2651 -2662
PubMed 23523385 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 9 8.18 9.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL517712 ATROPINE 4.0 1 9.92
CHEMBL1490 TRIHEXYPHENIDYL 4.0 1 8.82
CHEMBL1231 OXYBUTYNIN 4.0 1 8.70
CHEMBL1123 DICYCLOMINE 4.0 1 8.34
CHEMBL61946 CARAMIPHEN 2.0 1 8.14
CHEMBL1192807 1 8.07
CHEMBL9967 PIRENZEPINE 2.0 1 7.55
CHEMBL1192187 1 7.24
CHEMBL27673 METHOCTRAMINE 1 6.86

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL517712 ATROPINE Ki = 0.12 nM 9.92
CHEMBL1490 TRIHEXYPHENIDYL Ki = 1.5 nM 8.82
CHEMBL1231 OXYBUTYNIN Ki = 2.0 nM 8.70
CHEMBL1123 DICYCLOMINE Ki = 4.6 nM 8.34
CHEMBL61946 CARAMIPHEN Ki = 7.2 nM 8.14
CHEMBL1192807 Ki = 8.6 nM 8.07
CHEMBL9967 PIRENZEPINE Ki = 28.0 nM 7.55
CHEMBL1192187 Ki = 57.0 nM 7.24
CHEMBL27673 METHOCTRAMINE Ki = 137.0 nM 6.86