Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL2389280

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Staphylococcus aureus FabI using dodecenoyl ACP at pH 7.8
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Staphylococcus aureus
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Potential of lichen secondary metabolites against Plasmodium liver stage parasites with FAS-II as the potential target.
Lauinger IL, Vivas L, Perozzo R, Stairiker C, Tarun A, Zloh M, Zhang X, Xu H, Tonge PJ, Franzblau SG, Pham DH, Esguerra CV, Crawford AD, Maes L, Tasdemir D.
J Nat Prod (2013) 76 : 1064 -1070
PubMed 23806111 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 5.83 7.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL849 TRICLOSAN 4.0 1 7.60
CHEMBL463212 VULPINIC ACID 1 4.05
CHEMBL367881 (+)-USNIC ACID 1 -
CHEMBL176570 PSOROMIC ACID 1 -
CHEMBL1484978 EVERNIC ACID 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL849 TRICLOSAN IC50 = 25.0 nM 7.60
CHEMBL463212 VULPINIC ACID IC50 = 90000.0 nM 4.05
CHEMBL367881 (+)-USNIC ACID IC50 = 190000.0 nM -
CHEMBL176570 PSOROMIC ACID IC50 > 200000.0 nM -
CHEMBL1484978 EVERNIC ACID IC50 = 170000.0 nM -