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Assay Detail

CHEMBL2390268

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiplasmodial activity against Plasmodium falciparum by SYBR Green staining-based fluorescence assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Recent advances in malaria drug discovery.
Biamonte MA, Wanner J, Le Roch KG.
Bioorg Med Chem Lett (2013) 23 : 2829 -2843
PubMed 23587422 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 7.96 7.96

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL371405 MARIZOMIB 3.0 1 7.96

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL371405 MARIZOMIB EC50 = 11.0 nM 7.96