Assay Detail
Binding
CHEMBL2394914
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to sodium channel site 2 (unknown origin) by radioligand displacement assay
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 5.33 | 5.33 |
| IC50 | 1 | 5.28 | 5.28 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL439496 | VERATRIDINE | — | 2 | 5.33 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL439496 | VERATRIDINE | Ki | = | 4700.0 | nM | 5.33 |
| CHEMBL439496 | VERATRIDINE | IC50 | = | 5200.0 | nM | 5.28 |