Assay Detail
Binding
CHEMBL2395086
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Displacement of [3H]Glyburide from ATP-sensitive potassium channel in hamster pancreatic HIT-T15 cells after 2 hrs
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mesocricetus auratus |
| Cell Type | HIT-T15 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 9.19 | 9.19 |
| IC50 | 1 | 8.24 | 8.24 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL472 | GLYBURIDE | 4.0 | 2 | 9.19 |