Assay Detail
Binding
CHEMBL2396014
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in HEK293 cells after 1 to 1.5 hrs by scintillation counting analysis
4
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
An analysis of the synthetic tryptamines AMT and 5-MeO-DALT: emerging 'Novel Psychoactive Drugs'.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 7.38 | 7.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2391541 | — | — | 2 | 7.77 |
| CHEMBL30713 | — | — | 2 | 6.99 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2391541 | — | Ki | = | 17.0 | nM | 7.77 |
| CHEMBL2391541 | — | Ki | = | 16.98 | nM | 7.77 |
| CHEMBL30713 | — | Ki | = | 103.0 | nM | 6.99 |
| CHEMBL30713 | — | Ki | = | 102.33 | nM | 6.99 |