Assay Detail
Binding
CHEMBL2399302
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]DPDPE from delta opoid receptor in Dunkin-Hartley guinea pig brain after 2 hrs by liquid scintillation spectrometry
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cavia porcellus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Orally active opioid compounds from a non-poppy source.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 6.80 | 7.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL299031 | — | — | 1 | 7.22 |
| CHEMBL61630 | — | — | 1 | 6.81 |
| CHEMBL70 | MORPHINE | 4.0 | 1 | 6.38 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL299031 | — | Ki | = | 60.0 | nM | 7.22 |
| CHEMBL61630 | — | Ki | = | 155.0 | nM | 6.81 |
| CHEMBL70 | MORPHINE | Ki | = | 417.0 | nM | 6.38 |