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Assay Detail

CHEMBL2400447

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antioxidant activity assessed as DPPH radical scavenging activity after 30 mins by spectrophotometric analysis
26
Total Activities
26
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 3 — Cell-line / Tissue
Curated By Autocuration

Publication

Synthesis, antioxidant, and antimicrobial evaluation of some 2-arylbenzimidazole derivatives.
Zhou B, Li B, Yi W, Bu X, Ma L.
Bioorg Med Chem Lett (2013) 23 : 3759 -3763
PubMed 23711920 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 26 4.47 4.64

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2396683 1 4.64
CHEMBL2396701 1 4.58
CHEMBL2396684 1 4.57
CHEMBL2396697 1 4.52
CHEMBL2396685 1 4.50
CHEMBL2396700 1 4.48
CHEMBL2396699 1 4.47
CHEMBL242080 E319 1 4.44
CHEMBL2396698 1 4.40
CHEMBL2396656 1 4.38
CHEMBL2396692 1 4.24
CHEMBL2396696 1 -
CHEMBL2396695 1 -
CHEMBL2396694 1 -
CHEMBL2396693 1 -
CHEMBL2396691 1 -
CHEMBL2396690 1 -
CHEMBL2396689 1 -
CHEMBL2396688 1 -
CHEMBL2396687 1 -
CHEMBL1455814 1 -
CHEMBL379179 1 -
CHEMBL377740 1 -
CHEMBL2396686 1 -
CHEMBL203360 1 -
CHEMBL153535 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2396683 EC50 = 23000.0 nM 4.64
CHEMBL2396701 EC50 = 26000.0 nM 4.58
CHEMBL2396684 EC50 = 27000.0 nM 4.57
CHEMBL2396697 EC50 = 30000.0 nM 4.52
CHEMBL2396685 EC50 = 32000.0 nM 4.50
CHEMBL2396700 EC50 = 33000.0 nM 4.48
CHEMBL2396699 EC50 = 34000.0 nM 4.47
CHEMBL242080 E319 EC50 = 36000.0 nM 4.44
CHEMBL2396698 EC50 = 40000.0 nM 4.40
CHEMBL2396656 EC50 = 42000.0 nM 4.38
CHEMBL2396692 EC50 = 58000.0 nM 4.24
CHEMBL2396696 EC50 > 200000.0 nM -
CHEMBL2396695 EC50 > 200000.0 nM -
CHEMBL2396694 EC50 > 200000.0 nM -
CHEMBL2396693 EC50 > 200000.0 nM -
CHEMBL2396691 EC50 = 129000.0 nM -
CHEMBL2396690 EC50 > 200000.0 nM -
CHEMBL2396689 EC50 > 200000.0 nM -
CHEMBL2396688 EC50 > 200000.0 nM -
CHEMBL2396687 EC50 > 200000.0 nM -
CHEMBL1455814 EC50 > 200000.0 nM -
CHEMBL379179 EC50 > 200000.0 nM -
CHEMBL377740 EC50 > 200000.0 nM -
CHEMBL2396686 EC50 > 200000.0 nM -
CHEMBL203360 EC50 > 200000.0 nM -
CHEMBL153535 EC50 > 200000.0 nM -