Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL2403946

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [125I]substance P from human NK1 receptor expressed in CHO cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type CHO
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Substance-P receptor (CHEMBL249)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

2-[(3aR,4R,5S,7aS)-5-{(1S)-1-[3,5-bis(trifluoromethyl)phenyl]-2-hydroxyethoxy}-4-(2-methylphenyl)octahydro-2H-isoindol-2-yl]-1,3-oxazol-4(5H)-one: a potent human NK1 receptor antagonist with multiple clearance pathways.
Kassick AJ, Jiang J, Bunda J, Wilson D, Bao J, Lu H, Lin P, Ball RG, Doss GA, Tong X, Tsao KL, Wang H, Chicchi G, Karanam B, Tschirret-Guth R, Samuel K, Hora DF, Kumar S, Madeira M, Eng W, Hargreaves R, Purcell M, Gantert L, Cook J, DeVita RJ, Mills SG.
J Med Chem (2013) 56 : 5940 -5948
PubMed 23808489 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 10.22 10.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL447955 SERLOPITANT 3.0 1 10.22
CHEMBL2402572 1 10.22

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL447955 SERLOPITANT IC50 = 0.06 nM 10.22
CHEMBL2402572 IC50 = 0.06 nM 10.22