Assay Detail
Binding
CHEMBL2404253
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Induction of polyamine transport system-mediated compound uptake in mouse 4T1 cells after 72 hrs
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Cell Type | 4T1 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Development of polyamine transport ligands with improved metabolic stability and selectivity against specific human cancers.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.24 | 7.24 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2403110 | — | — | 1 | 7.24 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2403110 | — | IC50 | = | 57.6 | nM | 7.24 |