Assay Detail
Binding
CHEMBL2404442
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at adrenergic beta3 receptor (unknown origin) by PDSP assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Selectivity of phenothiazine cholinesterase inhibitors for neurotransmitter systems.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.69 | 5.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL394755 | — | — | 1 | 5.77 |
| CHEMBL240045 | — | — | 1 | 5.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL394755 | — | Ki | = | 1700.0 | nM | 5.77 |
| CHEMBL240045 | — | Ki | = | 2500.0 | nM | 5.60 |