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Assay Detail

CHEMBL2410405

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Influenza A virus A/Aichi/1968(H3N2) by firefly luciferase reporter gene assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Influenza A virus
Confidence 1 — Organism
Curated By Autocuration

Target

Influenza A virus (CHEMBL613740)
Type ORGANISM
Organism Influenza A virus

Publication

Synthesis and Metabolic Studies of Host Directed Inhibitors for Anti Viral Therapy.
Moore TW, Sana K, Yan D, Krumm SA, Thepchatri P, Snyder JP, Marengo J, Arrendale RF, Prussia AJ, Natchus MG, Liotta DC, Plemper RK, Sun A.
ACS Med Chem Lett (2013) 4 : 762 -767
PubMed 23956816 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 3 6.67 7.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1412578 1 7.30
CHEMBL1544917 1 6.04
CHEMBL2017637 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1412578 EC50 = 50.0 nM 7.30
CHEMBL1544917 EC50 = 920.0 nM 6.04
CHEMBL2017637 EC50 - -