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Assay Detail

CHEMBL2411599

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Functional
Antienteroviral activity against Human rhinovirus 63 infected in human HeLa Rh cells assessed as protection against virus-induced cytopathic effect after 2 to 3 days by MTS assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism rhinovirus A63
Cell Type HeLa Rh
Confidence 1 — Organism
Curated By Autocuration

Target

rhinovirus A63 (CHEMBL612478)
Type ORGANISM
Organism rhinovirus A63

Publication

Identification of a series of compounds with potent antiviral activity for the treatment of enterovirus infections.
MacLeod AM, Mitchell DR, Palmer NJ, Van de Poël H, Conrath K, Andrews M, Leyssen P, Neyts J.
ACS Med Chem Lett (2013) 4 : 585 -589
PubMed 24900715 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 7.65 8.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2407818 1 8.22
CHEMBL29609 PLECONARIL 2.0 1 7.07

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2407818 EC50 = 6.0 nM 8.22
CHEMBL29609 PLECONARIL EC50 = 85.0 nM 7.07