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Assay Detail

CHEMBL2411608

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Functional
Antienteroviral activity against Human rhinovirus 2 infected in human HeLa Rh cells assessed as protection against virus-induced cytopathic effect after 2 to 3 days by MTS assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism rhinovirus A2
Cell Type HeLa Rh
Confidence 1 — Organism
Curated By Autocuration

Target

rhinovirus A2 (CHEMBL612678)
Type ORGANISM
Organism rhinovirus A2

Publication

Identification of a series of compounds with potent antiviral activity for the treatment of enterovirus infections.
MacLeod AM, Mitchell DR, Palmer NJ, Van de Poël H, Conrath K, Andrews M, Leyssen P, Neyts J.
ACS Med Chem Lett (2013) 4 : 585 -589
PubMed 24900715 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 8.10 8.15

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL29609 PLECONARIL 2.0 1 8.15
CHEMBL2407818 1 8.05

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL29609 PLECONARIL EC50 = 7.0 nM 8.15
CHEMBL2407818 EC50 = 9.0 nM 8.05