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Assay Detail

CHEMBL2411684

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human HT-29 cells after 72 hrs by SRB assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HT-29
Confidence 1 — Organism
Curated By Autocuration

Target

HT-29 (CHEMBL384)
Type CELL-LINE
Organism Homo sapiens

Publication

Bioactive constituents of Indigofera spicata.
Bueno Pérez L, Li J, Lantvit DD, Pan L, Ninh TN, Chai HB, Soejarto DD, Swanson SM, Lucas DM, Kinghorn AD.
J Nat Prod (2013) 76 : 1498 -1504
PubMed 23895019 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 7.58 9.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL428647 PACLITAXEL 4.0 1 9.22
CHEMBL240545 ROTENOLONE 1 7.00
CHEMBL429023 ROTENONE 1 6.52
CHEMBL241806 TEPHROSIN 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL428647 PACLITAXEL IC50 = 0.6 nM 9.22
CHEMBL240545 ROTENOLONE IC50 = 100.0 nM 7.00
CHEMBL429023 ROTENONE IC50 = 300.0 nM 6.52
CHEMBL241806 TEPHROSIN IC50 > 10000.0 nM -