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Assay Detail

CHEMBL2416552

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to 5HT2C receptor (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

5-hydroxytryptamine receptor 2C (CHEMBL225)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Selective orexin receptor antagonists.
Lebold TP, Bonaventure P, Shireman BT.
Bioorg Med Chem Lett (2013) 23 : 4761 -4769
PubMed 23891187 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.92 5.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2111553 1 5.92

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2111553 Ki = 1200.0 nM 5.92