Assay Detail
Binding
CHEMBL2421968
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Competitive inhibition of human recombinant MAO-B expressed in insect cell microsomes using kynuramine as substrate by Lineweaver-Burk plot analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Subcellular | Microsome |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Selected furanochalcones as inhibitors of monoamine oxidase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.69 | 6.84 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2420790 | — | — | 1 | 6.84 |
| CHEMBL2420693 | — | — | 1 | 6.53 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2420790 | — | Ki | = | 144.0 | nM | 6.84 |
| CHEMBL2420693 | — | Ki | = | 294.0 | nM | 6.53 |