Assay Detail
Binding
CHEMBL2422672
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Inhibition of CDK9 (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Selectivity data: assessment, predictions, concordance, and implications.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.77 | 8.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1965660 | — | — | 1 | 8.00 |
| CHEMBL1967252 | — | — | 1 | 6.20 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 6.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1965660 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL1967252 | — | IC50 | = | 630.96 | nM | 6.20 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 794.33 | nM | 6.10 |