Assay Detail
Binding
CHEMBL2428681
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of trypsin amidolytic activity (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Thrombin inhibitory activity of some polyphenolic compounds.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.12 | 5.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL9509 | SILIBININ | 3.0 | 1 | 5.43 |
| CHEMBL50 | QUERCETIN | 3.0 | 1 | 4.81 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL9509 | SILIBININ | IC50 | = | 3700.0 | nM | 5.43 |
| CHEMBL50 | QUERCETIN | IC50 | = | 15400.0 | nM | 4.81 |