Assay Detail
Binding
CHEMBL2429348
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Binding affinity to CB1 receptor (unknown origin)
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Contributions of academic laboratories to the discovery and development of chemical biology tools.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 6.92 | 8.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL188 | WIN-552122 | — | 1 | 8.72 |
| CHEMBL408430 | — | — | 1 | 6.55 |
| CHEMBL306764 | — | — | 1 | 6.42 |
| CHEMBL497811 | — | — | 1 | 5.98 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL188 | WIN-552122 | Ki | = | 1.9 | nM | 8.72 |
| CHEMBL408430 | — | Ki | = | 280.0 | nM | 6.55 |
| CHEMBL306764 | — | Ki | = | 383.0 | nM | 6.42 |
| CHEMBL497811 | — | Ki | = | 1054.0 | nM | 5.98 |