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Assay Detail

CHEMBL2443919

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to sigma 2 receptor (unknown origin) by radioligand binding assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Discovery of an in vivo chemical probe of the lysine methyltransferases G9a and GLP.
Liu F, Barsyte-Lovejoy D, Li F, Xiong Y, Korboukh V, Huang XP, Allali-Hassani A, Janzen WP, Roth BL, Frye SV, Arrowsmith CH, Brown PJ, Vedadi M, Jin J.
J Med Chem (2013) 56 : 8931 -8942
PubMed 24102134 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 6.05 6.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2441082 1 6.05

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2441082 Ki = 900.0 nM 6.05