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Assay Detail

CHEMBL3054834

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Human poliovirus 1 strain Sabin infected African green monkey Vero76 cells assessed as reduction of virus-induced plaque reduction after 2 days by MTT assay
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Poliovirus 1
Cell Type Vero 76
Confidence 1 — Organism
Curated By Autocuration

Target

Poliovirus 1 (CHEMBL613556)
Type ORGANISM
Organism Poliovirus 1

Publication

Biological evaluation of novel 1,4-dithiine derivatives as potential antimicrobial agents
Bielenica A, Kossakowski J, Struga M, Dybaa I, La Colla P, Tamburini E, Loddo R
Med Chem Res (2011) 20 : 1411 -1420
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 8 4.75 4.75

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL98778 2'-ETHYNYL-D-CYTIDINE 1 4.75
CHEMBL2262347 1 -
CHEMBL2262145 1 -
CHEMBL2262345 1 -
CHEMBL2262344 1 -
CHEMBL2262348 1 -
CHEMBL2262359 1 -
CHEMBL2262357 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL98778 2'-ETHYNYL-D-CYTIDINE EC50 = 18000.0 nM 4.75
CHEMBL2262347 EC50 > 96000.0 nM -
CHEMBL2262145 EC50 > 100000.0 nM -
CHEMBL2262345 EC50 > 100000.0 nM -
CHEMBL2262344 EC50 > 100000.0 nM -
CHEMBL2262348 EC50 > 100000.0 nM -
CHEMBL2262359 EC50 > 100000.0 nM -
CHEMBL2262357 EC50 > 100000.0 nM -