Assay Detail
Binding
CHEMBL3056383
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Antagonist activity at alpha1D adrenoreceptor in Rattus norvegicus (rat) spleen
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Tissue | Spleen |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
(+)-Cyclazosin Derivatives as 1-Adrenoceptor Antagonists
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 6.86 | 6.86 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2261604 | (+)-CYCLAZOSIN | — | 1 | 6.86 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2261604 | (+)-CYCLAZOSIN | Kd | = | 138.04 | nM | 6.86 |