Assay Detail
Functional
CHEMBL3074875
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against Bovine viral diarrhea virus 1 infected bovine MDBK cells assessed as protection against virus-induced cytopathogenicity treated 1 hr after viral infection measured after 3-4 days by MTT method
23
Total Activities
23
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Bovine viral diarrhea virus 1 |
| Cell Type | MDBK |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Target
Bovine viral diarrhea virus 1 (CHEMBL612571) ↗| Type | ORGANISM |
| Organism | Bovine viral diarrhea virus 1 |
Publication
Syntheses and in vitro biological screening of 1-aryl-10H-[1,2,4]triazolo[3,4:3,4][1,2,4]triazino[5,6-b]indoles
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 23 | 4.87 | 5.75 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL418899 | 2'-B-METHYL-GUANOSINE | — | 1 | 5.75 |
| CHEMBL2296722 | — | — | 1 | 5.52 |
| CHEMBL2296717 | — | — | 1 | 4.16 |
| CHEMBL2296720 | — | — | 1 | 4.05 |
| CHEMBL2296721 | — | — | 1 | - |
| CHEMBL2296719 | — | — | 1 | - |
| CHEMBL2295851 | — | — | 1 | - |
| CHEMBL2296718 | — | — | 1 | - |
| CHEMBL2296716 | — | — | 1 | - |
| CHEMBL2296715 | — | — | 1 | - |
| CHEMBL2296714 | — | — | 1 | - |
| CHEMBL2296713 | — | — | 1 | - |
| CHEMBL2296712 | — | — | 1 | - |
| CHEMBL2296711 | — | — | 1 | - |
| CHEMBL2296710 | — | — | 1 | - |
| CHEMBL2296709 | — | — | 1 | - |
| CHEMBL2296708 | — | — | 1 | - |
| CHEMBL2296707 | — | — | 1 | - |
| CHEMBL2296706 | — | — | 1 | - |
| CHEMBL2296705 | — | — | 1 | - |
| CHEMBL2296704 | — | — | 1 | - |
| CHEMBL2296703 | — | — | 1 | - |
| CHEMBL2296702 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL418899 | 2'-B-METHYL-GUANOSINE | EC50 | = | 1800.0 | nM | 5.75 |
| CHEMBL2296722 | — | EC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL2296717 | — | EC50 | = | 69000.0 | nM | 4.16 |
| CHEMBL2296720 | — | EC50 | = | 90000.0 | nM | 4.05 |
| CHEMBL2296721 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296719 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2295851 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296718 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296716 | — | EC50 | > | 17000.0 | nM | - |
| CHEMBL2296715 | — | EC50 | > | 64000.0 | nM | - |
| CHEMBL2296714 | — | EC50 | > | 12000.0 | nM | - |
| CHEMBL2296713 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296712 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296711 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296710 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296709 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296708 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296707 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296706 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296705 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296704 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296703 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL2296702 | — | EC50 | > | 100000.0 | nM | - |