Assay Detail
Binding
CHEMBL3082947
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Inhibition of Bos taurus (bovine) pancrease carboxypeptidase A after 15 min
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bos taurus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Biological activity of tropolone.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.56 | 5.56 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL48310 | HINOKITIOL | — | 1 | 5.56 |
| CHEMBL121188 | TROPOLONE | — | 1 | 5.56 |
| CHEMBL415879 | PHENANTHROLINE | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL48310 | HINOKITIOL | IC50 | = | 2760.0 | nM | 5.56 |
| CHEMBL121188 | TROPOLONE | IC50 | = | 2730.0 | nM | 5.56 |
| CHEMBL415879 | PHENANTHROLINE | IC50 | = | 422000.0 | nM | - |