Assay Detail
Functional
CHEMBL3095696
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human NCI-H226 cells assessed as ATP level after 72 hrs by CellTiter-Glo assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NCI-H226 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
New synthetic enediynes and their conjugates may provide effective treatment for cancer.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 9.04 | 9.06 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3092453 | — | — | 1 | 9.06 |
| CHEMBL3092452 | — | — | 1 | 9.01 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3092453 | — | EC50 | = | 0.8729 | nM | 9.06 |
| CHEMBL3092452 | — | EC50 | = | 0.9859 | nM | 9.01 |