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Assay Detail

CHEMBL3097490

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H2]-25-hydroxycholesterol from N-terminal 6xHis-tagged human RORc ligand binding domain (241 to 486) expressed in bacterial expression system after 3 hrs by scintillation counting analysis
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Nuclear receptor ROR-gamma (CHEMBL1741186)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Structure-based design of substituted hexafluoroisopropanol-arylsulfonamides as modulators of RORc.
Fauber BP, de Leon Boenig G, Burton B, Eidenschenk C, Everett C, Gobbi A, Hymowitz SG, Johnson AR, Liimatta M, Lockey P, Norman M, Ouyang W, René O, Wong H.
Bioorg Med Chem Lett (2013) 23 : 6604 -6609
PubMed 24239186 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 29 6.26 7.47

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3094369 1 7.47
CHEMBL3094367 1 7.30
CHEMBL3094368 1 7.29
CHEMBL62136 T091317 1 7.22
CHEMBL3094366 1 6.72
CHEMBL2326845 1 6.61
CHEMBL3094384 1 6.48
CHEMBL3094379 1 6.33
CHEMBL3094378 1 6.29
CHEMBL3094365 1 6.28
CHEMBL3094372 1 6.28
CHEMBL3094370 1 6.13
CHEMBL3094380 1 6.05
CHEMBL205937 1 6.05
CHEMBL3094388 1 5.70
CHEMBL3094385 1 5.70
CHEMBL3094374 1 5.52
CHEMBL3094373 1 5.40
CHEMBL3094371 1 5.30
CHEMBL3094383 1 5.05
CHEMBL3094375 1 -
CHEMBL3094386 1 -
CHEMBL3094387 1 -
CHEMBL3094376 1 -
CHEMBL3094377 1 -
CHEMBL382792 1 -
CHEMBL389979 1 -
CHEMBL3094381 1 -
CHEMBL3094382 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3094369 IC50 = 34.0 nM 7.47
CHEMBL3094367 IC50 = 50.0 nM 7.30
CHEMBL3094368 IC50 = 51.0 nM 7.29
CHEMBL62136 T091317 IC50 = 60.0 nM 7.22
CHEMBL3094366 IC50 = 190.0 nM 6.72
CHEMBL2326845 IC50 = 245.0 nM 6.61
CHEMBL3094384 IC50 = 329.0 nM 6.48
CHEMBL3094379 IC50 = 467.0 nM 6.33
CHEMBL3094378 IC50 = 519.0 nM 6.29
CHEMBL3094365 IC50 = 520.0 nM 6.28
CHEMBL3094372 IC50 = 520.0 nM 6.28
CHEMBL3094370 IC50 = 748.0 nM 6.13
CHEMBL3094380 IC50 = 900.0 nM 6.05
CHEMBL205937 IC50 = 883.0 nM 6.05
CHEMBL3094388 IC50 = 2000.0 nM 5.70
CHEMBL3094385 IC50 = 2000.0 nM 5.70
CHEMBL3094374 IC50 = 3000.0 nM 5.52
CHEMBL3094373 IC50 = 4000.0 nM 5.40
CHEMBL3094371 IC50 = 5000.0 nM 5.30
CHEMBL3094383 IC50 = 9000.0 nM 5.05
CHEMBL3094375 IC50 > 10000.0 nM -
CHEMBL3094386 IC50 > 10000.0 nM -
CHEMBL3094387 IC50 > 10000.0 nM -
CHEMBL3094376 IC50 > 10000.0 nM -
CHEMBL3094377 IC50 > 10000.0 nM -
CHEMBL382792 IC50 > 10000.0 nM -
CHEMBL389979 IC50 > 10000.0 nM -
CHEMBL3094381 IC50 > 10000.0 nM -
CHEMBL3094382 IC50 > 10000.0 nM -