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Assay Detail

CHEMBL3101318

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of DOR (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Delta-type opioid receptor (CHEMBL236)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Imidazole-derived agonists for the neurotensin 1 receptor.
Hershberger PM, Hedrick MP, Peddibhotla S, Mangravita-Novo A, Gosalia P, Li Y, Gray W, Vicchiarelli M, Smith LH, Chung TD, Thomas JB, Caron MG, Pinkerton AB, Barak LS, Roth GP.
Bioorg Med Chem Lett (2014) 24 : 262 -267
PubMed 24332089 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.28 5.28

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL508044 1 5.28

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL508044 Ki = 5200.0 nM 5.28