Assay Detail
Functional
CHEMBL3101577
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Antiproliferative activity against human PC3 cells
28
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | PC-3 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
NAD-based inhibitors with anticancer potential.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 28 | 4.43 | 4.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3098170 | — | — | 1 | 4.96 |
| CHEMBL3098180 | — | — | 1 | 4.70 |
| CHEMBL2437262 | — | — | 1 | 4.21 |
| CHEMBL2437266 | — | — | 1 | 4.16 |
| CHEMBL2437258 | — | — | 1 | 4.10 |
| CHEMBL3098173 | — | — | 1 | - |
| CHEMBL3098172 | — | — | 1 | - |
| CHEMBL3098171 | — | — | 1 | - |
| CHEMBL3098169 | — | — | 1 | - |
| CHEMBL3098168 | — | — | 1 | - |
| CHEMBL3098167 | — | — | 1 | - |
| CHEMBL3098166 | — | — | 1 | - |
| CHEMBL3098165 | — | — | 1 | - |
| CHEMBL3098164 | — | — | 1 | - |
| CHEMBL3098163 | — | — | 1 | - |
| CHEMBL2437255 | — | — | 1 | - |
| CHEMBL3098175 | — | — | 1 | - |
| CHEMBL2437254 | — | — | 1 | - |
| CHEMBL2437265 | — | — | 1 | - |
| CHEMBL3098185 | — | — | 1 | - |
| CHEMBL2437269 | — | — | 1 | - |
| CHEMBL3098184 | — | — | 1 | - |
| CHEMBL2437273 | — | — | 1 | - |
| CHEMBL3098183 | — | — | 1 | - |
| CHEMBL2437272 | — | — | 1 | - |
| CHEMBL2437261 | — | — | 1 | - |
| CHEMBL3098182 | — | — | 1 | - |
| CHEMBL3098186 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3098170 | — | IC50 | = | 11000.0 | nM | 4.96 |
| CHEMBL3098180 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL2437262 | — | IC50 | = | 61000.0 | nM | 4.21 |
| CHEMBL2437266 | — | IC50 | = | 70000.0 | nM | 4.16 |
| CHEMBL2437258 | — | IC50 | = | 79000.0 | nM | 4.10 |
| CHEMBL3098173 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098172 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098171 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098169 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098168 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098167 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098166 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098165 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098164 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098163 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2437255 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098175 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2437254 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2437265 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098185 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2437269 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098184 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2437273 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098183 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2437272 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2437261 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098182 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098186 | — | IC50 | > | 100000.0 | nM | - |