Assay Detail
Functional
CHEMBL3106348
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human OX1 receptor overexpressed in CHO-RD-HGA16 cells assessed as calcium mobilization after 15 mins by fluorescence assay
28
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | RD-HGA16 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Truncated Orexin Peptides: Structure-Activity Relationship Studies.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 28 | 6.26 | 9.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL438925 | — | — | 1 | 9.66 |
| CHEMBL438397 | — | — | 1 | 8.08 |
| CHEMBL412459 | — | — | 1 | 7.19 |
| CHEMBL3103188 | — | — | 1 | 7.10 |
| CHEMBL3103893 | — | — | 1 | 6.84 |
| CHEMBL3103616 | — | — | 1 | 6.84 |
| CHEMBL3103189 | — | — | 1 | 6.67 |
| CHEMBL3105471 | — | — | 1 | 6.38 |
| CHEMBL3105470 | — | — | 1 | 6.31 |
| CHEMBL3105700 | — | — | 1 | 6.28 |
| CHEMBL3105701 | — | — | 1 | 6.27 |
| CHEMBL3105699 | — | — | 1 | 6.13 |
| CHEMBL3103894 | — | — | 1 | 6.06 |
| CHEMBL3105472 | — | — | 1 | 5.98 |
| CHEMBL3103895 | — | — | 1 | 5.95 |
| CHEMBL3103896 | — | — | 1 | 5.92 |
| CHEMBL3105698 | — | — | 1 | 5.87 |
| CHEMBL265424 | — | — | 1 | 5.86 |
| CHEMBL3103892 | — | — | 1 | 5.86 |
| CHEMBL3105702 | — | — | 1 | 5.81 |
| CHEMBL3103618 | — | — | 1 | 5.72 |
| CHEMBL3103187 | — | — | 1 | 5.72 |
| CHEMBL3105468 | — | — | 1 | 5.61 |
| CHEMBL3105473 | — | — | 1 | 5.51 |
| CHEMBL3105474 | — | — | 1 | 5.51 |
| CHEMBL3105703 | — | — | 1 | 5.51 |
| CHEMBL3105469 | — | — | 1 | 5.49 |
| CHEMBL3103186 | — | — | 1 | 5.24 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL438925 | — | EC50 | = | 0.22 | nM | 9.66 |
| CHEMBL438397 | — | EC50 | = | 8.29 | nM | 8.08 |
| CHEMBL412459 | — | EC50 | = | 64.0 | nM | 7.19 |
| CHEMBL3103188 | — | EC50 | = | 78.9 | nM | 7.10 |
| CHEMBL3103893 | — | EC50 | = | 143.0 | nM | 6.84 |
| CHEMBL3103616 | — | EC50 | = | 144.0 | nM | 6.84 |
| CHEMBL3103189 | — | EC50 | = | 212.0 | nM | 6.67 |
| CHEMBL3105471 | — | EC50 | = | 422.0 | nM | 6.38 |
| CHEMBL3105470 | — | EC50 | = | 493.0 | nM | 6.31 |
| CHEMBL3105700 | — | EC50 | = | 526.0 | nM | 6.28 |
| CHEMBL3105701 | — | EC50 | = | 535.0 | nM | 6.27 |
| CHEMBL3105699 | — | EC50 | = | 739.0 | nM | 6.13 |
| CHEMBL3103894 | — | EC50 | = | 865.0 | nM | 6.06 |
| CHEMBL3105472 | — | EC50 | = | 1040.0 | nM | 5.98 |
| CHEMBL3103895 | — | EC50 | = | 1130.0 | nM | 5.95 |
| CHEMBL3103896 | — | EC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL3105698 | — | EC50 | = | 1360.0 | nM | 5.87 |
| CHEMBL265424 | — | EC50 | = | 1380.0 | nM | 5.86 |
| CHEMBL3103892 | — | EC50 | = | 1370.0 | nM | 5.86 |
| CHEMBL3105702 | — | EC50 | = | 1560.0 | nM | 5.81 |
| CHEMBL3103618 | — | EC50 | = | 1910.0 | nM | 5.72 |
| CHEMBL3103187 | — | EC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL3105468 | — | EC50 | = | 2480.0 | nM | 5.61 |
| CHEMBL3105473 | — | EC50 | = | 3070.0 | nM | 5.51 |
| CHEMBL3105474 | — | EC50 | = | 3060.0 | nM | 5.51 |
| CHEMBL3105703 | — | EC50 | = | 3070.0 | nM | 5.51 |
| CHEMBL3105469 | — | EC50 | = | 3230.0 | nM | 5.49 |
| CHEMBL3103186 | — | EC50 | = | 5700.0 | nM | 5.24 |