Assay Detail
Binding
CHEMBL3119482
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Inhibition of pig heart MDH using chaperonin as substrate
36
Total Activities
36
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Sus scrofa |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
A biochemical screen for GroEL/GroES inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 36 | 4.64 | 5.26 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1632145 | — | — | 1 | 5.26 |
| CHEMBL3115910 | — | — | 1 | 4.72 |
| CHEMBL1376711 | — | — | 1 | 4.70 |
| CHEMBL3115915 | — | — | 1 | 4.30 |
| CHEMBL3115909 | — | — | 1 | 4.24 |
| CHEMBL3115926 | — | — | 1 | - |
| CHEMBL1411862 | — | — | 1 | - |
| CHEMBL3116089 | — | — | 1 | - |
| CHEMBL3116088 | — | — | 1 | - |
| CHEMBL3116087 | — | — | 1 | - |
| CHEMBL3116086 | — | — | 1 | - |
| CHEMBL3115929 | — | — | 1 | - |
| CHEMBL1775067 | — | — | 1 | - |
| CHEMBL3115928 | — | — | 1 | - |
| CHEMBL3115927 | — | — | 1 | - |
| CHEMBL3116090 | — | — | 1 | - |
| CHEMBL3115925 | — | — | 1 | - |
| CHEMBL3115908 | — | — | 1 | - |
| CHEMBL214344 | — | — | 1 | - |
| CHEMBL3115911 | — | — | 1 | - |
| CHEMBL2146958 | — | — | 1 | - |
| CHEMBL3115919 | — | — | 1 | - |
| CHEMBL3115913 | — | — | 1 | - |
| CHEMBL3115914 | — | — | 1 | - |
| CHEMBL3115916 | — | — | 1 | - |
| CHEMBL1713063 | — | — | 1 | - |
| CHEMBL3112623 | — | — | 1 | - |
| CHEMBL3115917 | — | — | 1 | - |
| CHEMBL3115918 | — | — | 1 | - |
| CHEMBL3115912 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1632145 | — | IC50 | = | 5500.0 | nM | 5.26 |
| CHEMBL3115910 | — | IC50 | = | 19000.0 | nM | 4.72 |
| CHEMBL1376711 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL3115915 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL3115909 | — | IC50 | = | 57000.0 | nM | 4.24 |
| CHEMBL3116087 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115920 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3116086 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115929 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL1775067 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115928 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115927 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3116090 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115925 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL1411862 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115924 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL1557710 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115923 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115922 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115921 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3116088 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3116089 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115926 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115908 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL214344 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115911 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL2146958 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115919 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115913 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115914 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115916 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL1713063 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3112623 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115917 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115918 | — | IC50 | > | 62500.0 | nM | - |
| CHEMBL3115912 | — | IC50 | > | 62500.0 | nM | - |