Assay Detail
Binding
CHEMBL3130639
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of HIV1 integrase/LEDGF-75 (unknown origin) interaction
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Inhibiting the HIV integration process: past, present, and the future.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 4.82 | 5.18 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1200748 | CARBIDOPA | 4.0 | 1 | 5.18 |
| CHEMBL1487 | ATORVASTATIN | 4.0 | 1 | 5.05 |
| CHEMBL3125907 | — | — | 1 | 4.60 |
| CHEMBL813 | EPROSARTAN | 4.0 | 1 | 4.43 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1200748 | CARBIDOPA | IC50 | = | 6540.0 | nM | 5.18 |
| CHEMBL1487 | ATORVASTATIN | IC50 | = | 8900.0 | nM | 5.05 |
| CHEMBL3125907 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL813 | EPROSARTAN | IC50 | = | 36850.0 | nM | 4.43 |